# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA254832 | 102, fendiline | IC50 | = | 7.8 | uM | ALA4817544 | 5.11 | nM | Homo sapiens | ||
2. | ALA4854753 | 22 | IC50 | = | 3.5 | uM | ALA4817544 | 5.46 | nM | Homo sapiens | ||
3. | ALA4859726 | 12h | IC50 | = | 3 | uM | ALA4817544 | 5.52 | nM | Homo sapiens | ||
4. | ALA4858481 | 12f | IC50 | = | 3.3 | uM | ALA4817544 | 5.48 | nM | Homo sapiens | ||
5. | ALA4849536 | 7 | IC50 | > | 30 | uM | ALA4817544 | nM | Homo sapiens | |||
6. | NI 42 | 15; Nl-42 | GI50 | = | 1 | uM | ALA4053040 | nM | Homo sapiens | |||
7. | ALA4586372 | 22a | IC50 | = | 274 | nM | ALA4412496 | 6.56 | nM | Homo sapiens | ||
8. | ALA3823303 | 5 | IC50 | = | 61 | nM | ALA4412496 | 7.21 | nM | Homo sapiens | ||
9. | ALA3764535 | 7 | RatioGI50 | = | 1500 | ALA3766762 | Homo sapiens | |||||
10. | Ulixertinib (BVD-523) | ULIXERTINIB | IC50 | = | 356 | nM | ALA4118533 | 6.45 | nM | Homo sapiens | ||
11. | ALA1614701 | AZD-6244 | IC50 | = | 117 | nM | ALA4118533 | 6.93 | nM | Homo sapiens | ||
12. | (5Z)-7-Oxozeaenol | 1, f152A1 | IC50 | = | 250 | nM | ALA4118533 | 6.60 | nM | Homo sapiens | ||
13. | ALA4127488 | 26 | IC50 | = | 2620 | nM | ALA4118533 | 5.58 | nM | Homo sapiens | ||
14. | N-{2-[(5-chloro-2-{[1-(2-methoxyethyl)-1H-pyrazol-4-yl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | 25 | IC50 | = | 318 | nM | ALA4118533 | 6.50 | nM | Homo sapiens | ||
15. | ALA3884293 | 9 | IC50 | = | 54 | nM | ALA4118533 | 7.27 | nM | Homo sapiens | ||
16. | ALA3884614 | 8 | IC50 | = | 213 | nM | ALA4118533 | 6.67 | nM | Homo sapiens | ||
17. | N-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamide | 5 | IC50 | = | 29 | nM | ALA4118533 | 7.54 | nM | Homo sapiens | ||
18. | ALA3884960 | 2 | IC50 | = | 294 | nM | ALA4118533 | 6.53 | nM | Homo sapiens | ||
19. | ALA5195618 | 44; SAH-SOS1A | EC50 | = | 100 | nM | ALA5150147 | 7.00 | nM | Homo sapiens | ||
20. | ALA5270178 | 5 | IC50 | = | 20 | uM | ALA5262102 | 4.70 | nM | Homo sapiens |