# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Khk-IN-1 | 8 | IC50 | > | 40 | uM | ALA2019661 | nM | Homo sapiens | |||
2. | ALA4094080 | 19 | INH | = | 17 | % | ALA4048663 | % | Homo sapiens | |||
3. | ALA1094408 | 49 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
4. | PF-04217903 | SID103905666 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
5. | SNS-032 (BMS-387032) | 21 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
6. | CH5183284 (Debio-1347) | 8; CH5183284; Debio 1347 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
7. | TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
8. | Alisertib (MLN8237) | 9, MLN-8237 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
9. | ASP3026 | ASP-3026 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
10. | ALA413 | Rapamycin | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
11. | Dabrafenib | 7, GSK2118436 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
12. | Abemaciclib | ABEMACICLIB | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
13. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
14. | ALA608533 | PKC-412 | Kd apparent | = | 1168 | nM | ALA3991839 | 5.93 | Active | nM | Homo sapiens | |
15. | Cobimetinib | 1, XL518, GDC-0973 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
16. | VX 702 | 5, VX-702 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
17. | CP-547632 | 1 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
18. | AT13148 | AT-13148 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
19. | R406 (free base) | 5, R-406 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens | ||
20. | GSK1070916 | GSK-1070916 | Kd apparent | > | 30000 | nM | ALA3991839 | Inactive | nM | Homo sapiens |