# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ARV-771 | 5 | DC50 | < | 1 | nM | ALA5246316 | nM | Homo sapiens | |||
2. | Mz1 | 1; MZ-1 | Emax | > | 90 | % | ALA5246305 | % | Homo sapiens | |||
3. | ARV-825 | 6; ARV-825 | DC50 | < | 1 | nM | ALA5246304 | nM | Homo sapiens | |||
4. | Mz1 | 1; MZ-1 | DC50 | < | 100 | nM | ALA5246304 | nM | Homo sapiens | |||
5. | ARV-825 | 6; ARV-825 | Kd | = | 28 | nM | ALA5246071 | 7.55 | nM | Homo sapiens | ||
6. | ARV-825 | 6; ARV-825 | Kd | = | 28 | nM | ALA5246070 | 7.55 | nM | Homo sapiens | ||
7. | ALA4850926 | 44 | IC50 | = | 11 | nM | ALA5245806 | 7.96 | nM | Homo sapiens | ||
8. | ALA4454646 | 59 | INH | = | 88 | % | ALA5245805 | % | Homo sapiens | |||
9. | ALA4454646 | 59 | IC50 | = | 5 | nM | ALA5245804 | 8.30 | nM | Homo sapiens | ||
10. | SB 202190 | 13 | IC50 | = | 3.4 | uM | ALA5245802 | 5.47 | nM | Homo sapiens | ||
11. | TG101209 | SID103904415 | IC50 | = | 130 | nM | ALA5245802 | 6.89 | nM | Homo sapiens | ||
12. | ALA5274032 | 19; MZ1 | Activity | = | 90 | % | ALA5245800 | % | Homo sapiens | |||
13. | dBET1 | 99 | Activity | = | 87 | % | ALA5245799 | % | Homo sapiens | |||
14. | ARV-825 | 6; ARV-825 | Kd | = | 20 | nM | ALA5245798 | 7.70 | nM | Homo sapiens | ||
15. | AZD-5153 | 103; AZD5153 | IC50 | = | 1.6 | nM | ALA5245796 | nM | Homo sapiens | |||
16. | AZD-5153 | 103; AZD5153 | IC50 | = | 5 | nM | ALA5245795 | 8.30 | nM | Homo sapiens | ||
17. | BI 2536 | 1 | IC50 | = | 25 | nM | ALA5245793 | 7.60 | nM | Homo sapiens | ||
18. | ALA5274937 | 7; MTI | IC50 | = | 3.1 | nM | ALA5245793 | 8.51 | nM | Homo sapiens | ||
19. | ALA5281214 | SJ995973; 26 | Emax | = | 87 | % | ALA5243428 | % | Homo sapiens | |||
20. | ALA5266070 | 34; BETd-246 | Emax | = | 63 | % | ALA5243427 | % | Homo sapiens |