| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2333445 | 1 | Activity | = | 100 | % | ALA2350108 | % | Homo sapiens | |||
| 2. |  ALA3220823 | 4g | Activity | = | 77 | % | ALA3223949 | % | Homo sapiens | |||
| 3. |  BAY-091 | EUB0001564 | % inhibition | 2.41 | % | ALA4887774 | Not Active | % | Homo sapiens | |||
| 4. |  ALA4580220 | EUB0000311 | % residual kinase activity | 78 | % | ALA4884220 | Not Active | % | Homo sapiens | |||
| 5. |  BAY-885 | BAY-885; 41 | % residual kinase activity | 96 | % | ALA4880955 | Not Active | % | Homo sapiens | |||
| 6. |  ALA4866102 | IIa | IC50 | = | 7058 | nM | ALA4832300 | 5.15 | nM | Homo sapiens | ||
| 7. |  ALA4856177 | 37d | Activity | < | 20 | % | ALA4830439 | % | Homo sapiens | |||
| 8. |  ALA4873571 | 13c | IC50 | > | 1000 | nM | ALA4823612 | nM | Homo sapiens | |||
| 9. |  ALA4859660 | I-9 | INH | = | 0 | % | ALA4804525 | % | Homo sapiens | |||
| 10. |  ALA4860979 | I-28 | INH | = | 0 | % | ALA4804525 | % | Homo sapiens | |||
| 11. |  ALA4855542 | I-13 | INH | = | 0 | % | ALA4804525 | % | Homo sapiens | |||
| 12. | ALA4859660 | I-9 | % inhibition | = | 9.5 | uM | ALA4804343 | Data is reported as I50 but values are consistent with % inhibition, changed for ChEMBL32 at suggestion of BZ | uM | Homo sapiens | ||
| 13. | ALA4860979 | I-28 | % inhibition | = | 8 | uM | ALA4804343 | Data is reported as I50 but values are consistent with % inhibition, changed for ChEMBL32 at suggestion of BZ | uM | Homo sapiens | ||
| 14. | ALA4855542 | I-13 | % inhibition | = | 16.7 | uM | ALA4804343 | Data is reported as I50 but values are consistent with % inhibition, changed for ChEMBL32 at suggestion of BZ | uM | Homo sapiens | ||
| 15. |  ALA4793380 | 17d | Activity | = | 39 | % | ALA4766691 | % | Homo sapiens | |||
| 16. |  Sorafenib | 5 | INH | = | 99.03 | % | ALA4735605 | % | Homo sapiens | |||
| 17. |  ALA4797840 | 1h | INH | = | -4 | % | ALA4735605 | % | Homo sapiens | |||
| 18. |  ALA4794578 | 7 | Activity | = | 95.88 | % | ALA4721295 | % | Homo sapiens | |||
| 19. |  ALA4750196 | 6g | Activity | = | 81.02 | % | ALA4721126 | % | Homo sapiens | |||
| 20. |  ALA4101882 | P-1 | IC50 | = | 194 | nM | ALA4050073 | 6.71 | nM | Homo sapiens |
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