# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4453882 | 3a; EC18 | EC50 | = | 21 | uM | ALA4433842 | 4.68 | nM | Mus musculus | ||
2. | ALA1253993 | 2 | INH | = | 35 | % | ALA1250983 | % | Mus musculus | |||
3. | ALA1253476 | (S)-6 | EC50 | = | 17.94 | uM | ALA1250984 | 4.75 | nM | Mus musculus | ||
4. | ALA1254085 | 3 | INH | = | 53 | % | ALA1250983 | % | Mus musculus | |||
5. | ALA1253478 | (R)-8 | INH | = | 60 | % | ALA1250983 | % | Mus musculus | |||
6. | ALA1253477 | 7 | INH | = | 82 | % | ALA1250983 | % | Mus musculus | |||
7. | ALA1253476 | (S)-6 | INH | = | 76 | % | ALA1250983 | % | Mus musculus | |||
8. | MEL57A | (R)-6 | INH | = | 27 | % | ALA1250983 | % | Mus musculus | |||
9. | ALA1254180 | (S)-5 | INH | = | 76 | % | ALA1250983 | % | Mus musculus | |||
10. | ALA1253992 | (R)-5 | INH | = | 63 | % | ALA1250983 | % | Mus musculus | |||
11. | ALA1254179 | (S)-4 | INH | = | 85 | % | ALA1250983 | % | Mus musculus | |||
12. | ALA1254086 | (R)-4 | INH | = | 85 | % | ALA1250983 | % | Mus musculus | |||
13. | Ivabradine | ivabradine | INH | = | 47 | % | ALA1250983 | % | Mus musculus | |||
14. | ALA1253479 | (S)-8 | INH | = | 93 | % | ALA1250983 | % | Mus musculus | |||
15. | ALA1254085 | 3 | EC50 | = | 5.6 | uM | ALA1250984 | 5.25 | nM | Mus musculus | ||
16. | ALA1253993 | 2 | EC50 | = | 2.31 | uM | ALA1250984 | 5.64 | nM | Mus musculus | ||
17. | ALA1254180 | (S)-5 | EC50 | = | 31.27 | uM | ALA1250984 | 4.50 | nM | Mus musculus | ||
18. | MEL57A | (R)-6 | EC50 | = | 0.6 | uM | ALA1250984 | 6.22 | nM | Mus musculus | ||
19. | Ivabradine | ivabradine | EC50 | = | 4.5 | uM | ALA1250984 | 5.35 | nM | Mus musculus | ||
20. | ALA1253992 | (R)-5 | EC50 | = | 9.41 | uM | ALA1250984 | 5.03 | nM | Mus musculus |