# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | zatebradine | Zetebradine | INH | = | 59 | % | ALA4433868 | % | Homo sapiens | |||
2. | ALA4453882 | 3a; EC18 | EC50 | = | 3.98 | uM | ALA4433840 | 5.40 | nM | Homo sapiens | ||
3. | ALA4435474 | 3g | INH | = | 30 | % | ALA4433839 | % | Homo sapiens | |||
4. | ALA4476524 | 3f | INH | = | 4 | % | ALA4433839 | % | Homo sapiens | |||
5. | ALA4449749 | 3e | INH | = | 64 | % | ALA4433839 | % | Homo sapiens | |||
6. | ALA4464995 | 3d | INH | = | 48 | % | ALA4433839 | % | Homo sapiens | |||
7. | ALA4449514 | 3c | INH | = | 47 | % | ALA4433839 | % | Homo sapiens | |||
8. | ALA4460609 | 3b | INH | = | 21 | % | ALA4433839 | % | Homo sapiens | |||
9. | EC18 | (+)-3a; (+)-EC18 | INH | = | 45 | % | ALA4433839 | % | Homo sapiens | |||
10. | EC18 | (+)-3a; (+)-EC18 | INH | = | 46 | % | ALA4433839 | % | Homo sapiens | |||
11. | ALA4453882 | 3a; EC18 | INH | = | 59 | % | ALA4433839 | % | Homo sapiens | |||
12. | ALA4440935 | 29; CYM-51317 | INH | < | 25 | % | ALA4424289 | % | Homo sapiens | |||
13. | ALA4459625 | 36 | INH | 0 | ALA4424289 | Not Determined | % | Homo sapiens | ||||
14. | ALA4434885 | 35 | INH | 0 | ALA4424289 | Not Determined | % | Homo sapiens | ||||
15. | ALA4576339 | 34 | INH | < | 25 | % | ALA4424289 | % | Homo sapiens | |||
16. | 5-Chloro-4-(4-chloro-1-methyl-1H-pyrazol-5-yl)-N-((3S,4S,6S)-4-(3,4-difluorophenyl)-6-(2-(methylamino)-2-oxoethyl)piperidin-3-yl)furan-2-carboxamide | E22 | INH | 0 | ALA4407446 | Not Active | % | Homo sapiens | ||||
17. | AZD5718 | 12; AZD5718 | IC50 | > | 32 | uM | ALA4393840 | nM | Homo sapiens | |||
18. | ALA4474619 | 11 | IC50 | > | 32 | uM | ALA4393840 | nM | Homo sapiens | |||
19. | CCT245737 | CCT245737 | IC50 | > | 10 | uM | ALA4706995 | nM | Homo sapiens | |||
20. | ALA4528928 | 4i | INH | 0 | ALA4351291 | Not Active | % | Homo sapiens |