# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Tazobactam acid | 2 Tazobactam | IC50 | = | 0.08 | uM | ALA1262649 | 7.10 | nM | Klebsiella pneumoniae | ||
2. | clavulanic acid | Clavulanic acid | IC50 | = | 1.72 | uM | ALA1262649 | 5.76 | nM | Klebsiella pneumoniae | ||
3. | Cefotaxime acid | cefotaxime | Kcat/Km | 0 | ALA1262647 | Not Determined | Klebsiella pneumoniae | |||||
4. | Ceftazidime (containing approximately 10% sodium carbonate) | CAZ | Kcat/Km | 0 | ALA1262647 | Not Determined | Klebsiella pneumoniae | |||||
5. | ALA617 | Cephalothin | Kcat/Km | = | 0.3 | /uM/s | ALA1262647 | /uM/s | Klebsiella pneumoniae | |||
6. | Piperacillin | Piperacillin | Kcat/Km | = | 44.6 | /uM/s | ALA1262647 | /uM/s | Klebsiella pneumoniae | |||
7. | ticarcillin | ticarcillin | Kcat/Km | = | 35.5 | /uM/s | ALA1262647 | /uM/s | Klebsiella pneumoniae | |||
8. | Amoxicillin | amoxicilln | Kcat/Km | = | 226 | /uM/s | ALA1262647 | /uM/s | Klebsiella pneumoniae | |||
9. | penicillin G | Benzylpenicillin | Kcat/Km | = | 286.2 | /uM/s | ALA1262647 | /uM/s | Klebsiella pneumoniae | |||
10. | Cefotaxime acid | cefotaxime | Kcat | < | 0.1 | /s | ALA1262645 | /s | Klebsiella pneumoniae | |||
11. | Ceftazidime (containing approximately 10% sodium carbonate) | CAZ | Kcat | < | 0.1 | /s | ALA1262645 | /s | Klebsiella pneumoniae | |||
12. | ALA617 | Cephalothin | Kcat | = | 38 | /s | ALA1262645 | /s | Klebsiella pneumoniae | |||
13. | Piperacillin | Piperacillin | Kcat | = | 1918 | /s | ALA1262645 | /s | Klebsiella pneumoniae | |||
14. | ticarcillin | ticarcillin | Kcat | = | 1279 | /s | ALA1262645 | /s | Klebsiella pneumoniae | |||
15. | Amoxicillin | amoxicilln | Kcat | = | 5876 | /s | ALA1262645 | /s | Klebsiella pneumoniae | |||
16. | penicillin G | Benzylpenicillin | Kcat | = | 5438 | /s | ALA1262645 | /s | Klebsiella pneumoniae | |||
17. | Cefotaxime acid | cefotaxime | Km | 0 | ALA1262645 | Not Determined | Klebsiella pneumoniae | |||||
18. | Ceftazidime (containing approximately 10% sodium carbonate) | CAZ | Km | 0 | ALA1262645 | Not Determined | Klebsiella pneumoniae | |||||
19. | ALA617 | Cephalothin | Km | = | 141 | uM | ALA1262645 | nM | Klebsiella pneumoniae | |||
20. | Piperacillin | Piperacillin | Km | = | 43 | uM | ALA1262645 | nM | Klebsiella pneumoniae |