# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5266562 | 43 | IC50 | = | 0.49 | uM | ALA5237563 | 6.31 | nM | Homo sapiens | ||
2. | MS049 | 17; MS049 | Kd | = | 87 | nM | ALA5214691 | 7.06 | nM | Homo sapiens | ||
3. | MS049 | 17; MS049 | dTm | = | 11.3 | K | ALA5214690 | K | Homo sapiens | |||
4. | MS023 | 3 | Kd | = | 6 | nM | ALA5214676 | 8.22 | nM | Homo sapiens | ||
5. | A 366 | 12, A-366 | EC50 | > | 50 | uM | ALA5214737 | nM | Homo sapiens | |||
6. | OICR-9429 | 16d; OICR-9429 | % activity remaining | > | 90 | % | ALA5213727 | % | Homo sapiens | |||
7. | MS049 | 17; MS049 | IC50 | = | 43 | nM | ALA5210604 | 7.37 | nM | Homo sapiens | ||
8. | MS023 | 3 | IC50 | = | 4 | nM | ALA5210601 | 8.40 | nM | Homo sapiens | ||
9. | MS049 | 17; MS049 | IC50 | = | 970 | nM | ALA5210296 | 6.01 | nM | Homo sapiens | ||
10. | MS023 | 3 | IC50 | = | 56 | nM | ALA5210294 | 7.25 | nM | Homo sapiens | ||
11. | ALA5195436 | 9; MS159 | INH | 0 | ALA5141723 | NA | % | Homo sapiens | ||||
12. | ALA5173678 | 12h; EML981 | IC50 | = | 1.75 | uM | ALA5138948 | 5.76 | nM | Homo sapiens | ||
13. | ALA5191769 | 12g; EML982 | IC50 | = | 4.34 | uM | ALA5138948 | 5.36 | nM | Homo sapiens | ||
14. | ALA5202088 | 12f; EML980 | IC50 | = | 22.7 | uM | ALA5138948 | 4.64 | nM | Homo sapiens | ||
15. | ALA5186617 | 12e; EML979 | IC50 | = | 35.6 | uM | ALA5138948 | 4.45 | nM | Homo sapiens | ||
16. | ALA5180108 | 12d; EML978 | IC50 | = | 47 | uM | ALA5138948 | 4.33 | nM | Homo sapiens | ||
17. | ALA5206272 | 12c; EML736 | IC50 | > | 100 | uM | ALA5138948 | nM | Homo sapiens | |||
18. | ALA5170047 | 12b; EML709 | IC50 | > | 100 | uM | ALA5138948 | nM | Homo sapiens | |||
19. | ALA5199380 | 12a; EML734 | IC50 | = | 72.77 | uM | ALA5138948 | 4.14 | nM | Homo sapiens | ||
20. | ALA5197421 | 74 | IC50 | = | 90 | nM | ALA5138254 | 7.05 | nM | Homo sapiens |