# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ketohexokinase inhibitor 1 | 51 | IC50 | = | 10 | nM | ALA5150316 | 8.00 | nM | Homo sapiens | ||
2. | Ketohexokinase inhibitor 1 | 51 | IC50 | = | 0.014 | uM | ALA4344288 | 7.85 | nM | Homo sapiens | ||
3. | ALA4070442 | 12 | IC50 | = | 0.45 | uM | ALA4344288 | 6.35 | nM | Homo sapiens | ||
4. | 3-(Trifluoromethyl)quinoxalin-2(1H)-one | SID26667233 | Kd | = | 44 | uM | ALA4344289 | 4.36 | nM | Homo sapiens | ||
5. | 3-(Trifluoromethyl)quinoxalin-2(1H)-one | SID26667233 | IC50 | = | 319 | uM | ALA4344288 | nM | Homo sapiens | |||
6. | ALA1500542 | SID14726509 | Kd | = | 62 | uM | ALA4344289 | 4.21 | nM | Homo sapiens | ||
7. | ALA1500542 | SID14726509 | IC50 | = | 319 | uM | ALA4344288 | nM | Homo sapiens | |||
8. | Ketohexokinase inhibitor 1 | 51 | INH | 0 | ALA4676081 | Active | % | Homo sapiens | ||||
9. | Ketohexokinase inhibitor 1 | 51 | Ki | = | 4.53 | nM | ALA4676080 | 8.34 | nM | Homo sapiens | ||
10. | Ketohexokinase inhibitor 1 | 51 | INH | 0 | ALA4676079 | Not Active | % | Homo sapiens | ||||
11. | Ketohexokinase inhibitor 1 | 51 | INH | 0 | ALA4676074 | Active | % | Homo sapiens | ||||
12. | Ketohexokinase inhibitor 1 | 51 | INH | 0 | ALA4676073 | Active | % | Homo sapiens | ||||
13. | Ketohexokinase inhibitor 1 | 51 | IC50 | = | 0.17 | uM | ALA4676065 | 6.77 | nM | Homo sapiens | ||
14. | Ketohexokinase inhibitor 1 | 51 | IC50 | = | 0.028 | uM | ALA4676064 | 7.55 | nM | Homo sapiens | ||
15. | Ketohexokinase inhibitor 1 | 51 | IC50 | = | 0.01 | uM | ALA4676055 | 8.00 | nM | Homo sapiens | ||
16. | ALA4782925 | 7 | IC50 | = | 0.014 | uM | ALA4676055 | 7.85 | nM | Homo sapiens | ||
17. | ALA4754053 | 6 | IC50 | = | 0.001 | uM | ALA4676055 | 9.00 | nM | Homo sapiens | ||
18. | ALA4760155 | 4 | IC50 | = | 0.14 | uM | ALA4676054 | 6.85 | nM | Homo sapiens | ||
19. | ALA4798024 | 3 | IC50 | = | 0.47 | uM | ALA4676054 | 6.33 | nM | Homo sapiens | ||
20. | ALA4762437 | 2 | IC50 | = | 0.41 | uM | ALA4676054 | 6.39 | nM | Homo sapiens |