| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 34 | nM | ALA4337459 | 7.47 | nM | Rattus norvegicus | ||
| 2. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Intrinsic activity | = | 0.4 | ALA4337456 | Rattus norvegicus | |||||
| 3. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | pEC50 | = | 6.8 | ALA4337455 | 6.80 | nM | Rattus norvegicus | |||
| 4. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Intrinsic activity | = | -0.2 | ALA4337454 | Rattus norvegicus | |||||
| 5. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | pEC50 | = | 4.3 | ALA4337453 | 4.30 | nM | Rattus norvegicus | |||
| 6. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | pKi | = | 5.71 | ALA4337440 | 5.71 | nM | Rattus norvegicus | |||
| 7. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.2 | /min | ALA4337437 | /min | Rattus norvegicus | |||
| 8. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.13 | /min | ALA4337434 | /min | Rattus norvegicus | |||
| 9. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | t1/2 | = | 6.6 | min | ALA4337431 | hr | Rattus norvegicus | |||
| 10. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.11 | /min | ALA4337428 | /min | Rattus norvegicus | |||
| 11. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.003 | /min/nM | ALA4337425 | /min/nM | Rattus norvegicus | |||
| 12. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.205 | /min | ALA4337422 | /min | Rattus norvegicus | |||
| 13. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 34 | nM | ALA4337419 | 7.47 | nM | Rattus norvegicus | ||
| 14. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 21.8 | nM | ALA4337416 | 7.66 | nM | Rattus norvegicus | ||
| 15. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 22.2 | nM | ALA4337413 | 7.65 | nM | Rattus norvegicus | ||
| 16. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Bmax | = | 2455 | disintegrations/minute | ALA4337413 | disintegrations/minute | Rattus norvegicus | |||
| 17. |  ALA4445423 | 49 | Intrinsic activity | = | 0.92 | ALA4337409 | Rattus norvegicus | |||||
| 18. |  ALA4543119 | 48 | Intrinsic activity | = | 0.75 | ALA4337409 | Rattus norvegicus | |||||
| 19. |  ALA4439142 | 46; UR-DEBa176 | Intrinsic activity | = | 0.68 | ALA4337409 | Rattus norvegicus | |||||
| 20. |  ALA4443126 | 45 | Intrinsic activity | = | 0.11 | ALA4337409 | Rattus norvegicus |
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