| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Thioperamide | Thioperamide | pKi | = | 7.3 | ALA2154955 | 7.30 | nM | Rattus norvegicus | |||
| 2. |  JNJ-39758979 | 5, JNJ 39758979 | pA2 | = | 7.2 | ALA3241492 | 7.20 | nM | Rattus norvegicus | |||
| 3. | JNJ-39758979 | 5, JNJ 39758979 | Ki | = | 188 | nM | ALA3241491 | 6.73 | nM | Rattus norvegicus | ||
| 4. | JNJ-39758979 | 5, JNJ 39758979 | Ki | = | 188 | nM | ALA3626552 | 6.73 | nM | Rattus norvegicus | ||
| 5. |  adriforant | 13, PF-3893787 | pKi | = | 7.91 | ALA3626545 | 7.91 | nM | Rattus norvegicus | |||
| 6. |  Histamine, Free Base | histamine | Ki | = | 136 | nM | ALA3626540 | 6.87 | nM | Rattus norvegicus | ||
| 7. |  ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 34 | nM | ALA4337459 | 7.47 | nM | Rattus norvegicus | ||
| 8. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Intrinsic activity | = | 0.4 | ALA4337456 | Rattus norvegicus | |||||
| 9. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | pEC50 | = | 6.8 | ALA4337455 | 6.80 | nM | Rattus norvegicus | |||
| 10. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Intrinsic activity | = | -0.2 | ALA4337454 | Rattus norvegicus | |||||
| 11. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | pEC50 | = | 4.3 | ALA4337453 | 4.30 | nM | Rattus norvegicus | |||
| 12. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | pKi | = | 5.71 | ALA4337440 | 5.71 | nM | Rattus norvegicus | |||
| 13. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.2 | /min | ALA4337437 | /min | Rattus norvegicus | |||
| 14. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.13 | /min | ALA4337434 | /min | Rattus norvegicus | |||
| 15. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | t1/2 | = | 6.6 | min | ALA4337431 | hr | Rattus norvegicus | |||
| 16. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.11 | /min | ALA4337428 | /min | Rattus norvegicus | |||
| 17. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.003 | /min/nM | ALA4337425 | /min/nM | Rattus norvegicus | |||
| 18. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | K | = | 0.205 | /min | ALA4337422 | /min | Rattus norvegicus | |||
| 19. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 34 | nM | ALA4337419 | 7.47 | nM | Rattus norvegicus | ||
| 20. | ALA4515149 | [3H]-46; [3H]UR-DEBa176 | Kd | = | 21.8 | nM | ALA4337416 | 7.66 | nM | Rattus norvegicus |
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