| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Probenecid | probenecid | Ki | = | 221 | uM | ALA1908125 | nM | Homo sapiens | |||
| 2. |  Diclofenac | 25 (Diclofenac) | Ki | = | 52 | uM | ALA1908125 | 4.28 | nM | Homo sapiens | ||
| 3. |  ALA408 | Troglitazone | Vmax | = | 12 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 4. |  Naltrexone | naltrexone | Vmax | = | 2 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 5. |  nalorphine | nalorphine | Vmax | = | 2 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 6. |  Mycophenolic acid | MPA | Vmax | = | 336 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 7. |  ALA1329 | Morphine 3-Glucuronide | Vmax | = | 4.5 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 8. |  α-Hydroxy Tamoxifen | cis-Hydroxy-tamoxifen | Vmax | = | 166 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 9. | α-Hydroxy Tamoxifen | cis-Hydroxy-tamoxifen | Vmax | = | 291 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 10. |  Ezetimibe | 2 (-) | Vmax | = | 710 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 11. |  Etoposide | VP-16 | Vmax | = | 267 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 12. |  ALA837 | 44 | Vmax | = | 134 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 13. |  ALA2303616 | Entacapone (glucuronidation 1) | Vmax | = | 5 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 14. |  ALA2303615 | Entacapone (3-O-glucuronidation) | Vmax | = | 4 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 15. |  Ethinyl Estradiol | 17 alpha-ethynyl E2 | Vmax | = | 59 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 16. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | Vmax | = | 650 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 17. |  (1S,2S,6R,14R,15S,16R)-5-(cyclopropylmethyl)-16-[(2S)-2-hydroxy-3,3-dimethylbutan-2-yl]-15-methoxy-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-trien-11-ol | 1a | Vmax | = | 555 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 18. | (1S,2S,6R,14R,15S,16R)-5-(cyclopropylmethyl)-16-[(2S)-2-hydroxy-3,3-dimethylbutan-2-yl]-15-methoxy-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-trien-11-ol | 1a | Vmax | = | 2500 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 19. |  4-Acetamidophenol | 1 | Vmax | = | 1300 | pmol/min/mg protein | ALA1908113 | pmol/min/mg protein | Homo sapiens | |||
| 20. | ALA408 | Troglitazone | Km | = | 58 | uM | ALA1908113 | nM | Homo sapiens |
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