Activities

#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	ALA2036782	8c	IC50	=	0.2	uM	ALA2039636	6.70		nM	Rattus norvegicus
2.	N-[2-[(3S)-3-[[cis-4-hydroxy-4-(5-pyrimidin-2-yl-2-pyridyl)cyclohexyl]amino]pyrrolidin-1-yl]-2-oxo-ethyl]-3-(trifluoromethyl)benzamide	17, INCB3284	IC50	=	13	nM	ALA2032547	7.89		nM	Rattus norvegicus
3.	N-[2-[(3S)-3-[[cis-4-hydroxy-4-(5-pyrimidin-2-yl-2-pyridyl)cyclohexyl]amino]pyrrolidin-1-yl]-2-oxo-ethyl]-3-(trifluoromethyl)benzamide	17, INCB3284	IC50	=	2.8	nM	ALA2032549	8.55		nM	Rattus norvegicus
4.	ALA3770912	2f	IC50	=	1.3	nM	ALA3772539	8.89		nM	Rattus norvegicus
5.	ALA1688889	17	IC50	=	10	uM	ALA1693911	5.00		nM	Rattus norvegicus
6.	ALA1688888	13	IC50		0		ALA1693911		Not Determined		Rattus norvegicus
7.	ALA1683074	19	IC50	=	2.9	nM	ALA1685783	8.54		nM	Rattus norvegicus
8.	ALA1289316	21, INCB-3344	IC50	=	7.3	uM	ALA1291446	5.14		nM	Rattus norvegicus