# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4875978 | ML-SI1; racemic mixture(55:45) | IC50 | 0 | ALA4819517 | Not Active | Homo sapiens | |||||
2. | ALA4856175 | (+/-)-trans-ML-SI3 | IC50 | = | 17 | uM | ALA4819517 | 4.77 | nM | Homo sapiens | ||
3. | ALA4847300 | 18 | INH | 0 | ALA4819514 | Active | % | Homo sapiens | ||||
4. | ALA4875978 | ML-SI1; racemic mixture(55:45) | INH | 0 | ALA4819514 | Not Active | % | Homo sapiens | ||||
5. | ALA4856175 | (+/-)-trans-ML-SI3 | INH | 0 | ALA4819514 | Not Active | % | Homo sapiens | ||||
6. | ALA4856175 | (+/-)-trans-ML-SI3 | INH | 0 | ALA4819514 | Active | % | Homo sapiens | ||||
7. | ALA4875551 | 31 | EC50 | 0 | ALA4819513 | Not Active | Homo sapiens | |||||
8. | ALA4855589 | 26 | EC50 | 0 | ALA4819513 | Not Active | Homo sapiens | |||||
9. | ALA4856325 | 25 | EC50 | 0 | ALA4819513 | Not Active | Homo sapiens | |||||
10. | ALA4858349 | 20 | EC50 | 0 | ALA4819513 | Not Active | Homo sapiens | |||||
11. | ALA4847300 | 18 | EC50 | 0 | ALA4819513 | Not Active | Homo sapiens | |||||
12. | ALA4856175 | (+/-)-trans-ML-SI3 | EC50 | 0 | ALA4819513 | Not Active | Homo sapiens | |||||
13. | ALA4856175 | (+/-)-trans-ML-SI3 | EC50 | 0 | ALA4819513 | Not Active | Homo sapiens | |||||
14. | ALA4851134 | 28 | EC50 | = | 9.5 | uM | ALA4819513 | 5.02 | nM | Homo sapiens | ||
15. | ALA4874310 | 27 | EC50 | = | 20.7 | uM | ALA4819513 | 4.68 | nM | Homo sapiens | ||
16. | ALA4856363 | 24 | EC50 | = | 5.4 | uM | ALA4819513 | 5.27 | nM | Homo sapiens | ||
17. | ALA4870275 | 23 | EC50 | = | 5.8 | uM | ALA4819513 | 5.24 | nM | Homo sapiens | ||
18. | ALA4855846 | 22 | EC50 | = | 14.6 | uM | ALA4819513 | 4.84 | nM | Homo sapiens | ||
19. | ALA4849322 | 21 | EC50 | = | 9.5 | uM | ALA4819513 | 5.02 | nM | Homo sapiens | ||
20. | ALA4857820 | 17 | EC50 | = | 8.5 | uM | ALA4819513 | 5.07 | nM | Homo sapiens |