# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | CLK-IN-T3 | EUB0000321 | IC50 | > | 10 | uM | ALA5213250 | nM | Homo sapiens | |||
2. | CLK-IN-T3 | EUB0000321 | % of control | = | 4.9 | % | ALA5213249 | % | Homo sapiens | |||
3. | LDC1267 | 7; LDC1267 | Kd | = | 124 | nM | ALA5212916 | 6.91 | nM | Homo sapiens | ||
4. | LDC1267 | 7; LDC1267 | % of control | < | 10 | % | ALA5212915 | % | Homo sapiens | |||
5. | GW843682X | 2 | % of control | = | 0.5 | % | ALA5213203 | % | Homo sapiens | |||
6. | ALA4557026 | EUB0000700 | % of control | = | 17.6 | % | ALA5213292 | % | Homo sapiens | |||
7. | BAY-985 | 34; BAY-985 | IC50 | > | 20 | uM | ALA5213273 | nM | Homo sapiens | |||
8. | BAY-985 | 34; BAY-985 | % of control | = | 8.5 | % | ALA5213272 | % | Homo sapiens | |||
9. | BAY-985 | 34; BAY-985 | IC50 | = | 847 | nM | ALA5213271 | 6.07 | nM | Homo sapiens | ||
10. | ALA4538591 | 36; BAY-440 | % of control | = | 1.8 | % | ALA5213295 | % | Homo sapiens | |||
11. | ALA4530401 | EUB0000704 | % of control | = | 25.2 | % | ALA5213470 | % | Homo sapiens | |||
12. | BI 99179 | 13, BI-99179 | % of control | = | 16 | % | ALA5213851 | % | Homo sapiens | |||
13. | ALA2381342 | BIX02189 | IC50 | = | 1.5 | nM | ALA5166121 | 8.82 | nM | Homo sapiens | ||
14. | ALA5193786 | 34b | Kd | = | 2.8 | nM | ALA5166111 | 8.55 | nM | Homo sapiens | ||
15. | ALA5190298 | 22 | INH | = | 78 | % | ALA5149686 | % | Homo sapiens | |||
16. | ALA4550647 | 31 | Activity | <= | 1 | % | ALA4478333 | % | Homo sapiens | |||
17. | ALA4571241 | 9im | Kd | = | 38 | nM | ALA4426908 | 7.42 | nM | Homo sapiens | ||
18. | ALA4458435 | 23; PF-06700841 | INH | = | 70 | % | ALA4411560 | % | Homo sapiens | |||
19. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405446 | % | Homo sapiens | |||
20. | ALA4447797 | 28 | Activity | 0 | ALA4394536 | Active | Homo sapiens |