# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ARV-771 | 5 | Emax | > | 90 | % | ALA5246317 | % | Homo sapiens | |||
2. | ARV-771 | 5 | DC50 | < | 1 | nM | ALA5246314 | nM | Homo sapiens | |||
3. | ALA5283149 | 43 | Kd | = | 180 | nM | ALA5243397 | 6.75 | nM | Homo sapiens | ||
4. | Mz1 | 1; MZ-1 | Kd | = | 740 | nM | ALA5243397 | 6.13 | nM | Homo sapiens | ||
5. | ARV-771 | 5 | DC50 | < | 5 | nM | ALA5243380 | nM | Homo sapiens | |||
6. | ARV-771 | 5 | DC50 | < | 5 | nM | ALA5243379 | nM | Homo sapiens | |||
7. | ARV-771 | 5 | DC50 | < | 5 | nM | ALA5243378 | nM | Homo sapiens | |||
8. | Mz1 | 1; MZ-1 | Kd | = | 115 | nM | ALA5243375 | 6.94 | nM | Homo sapiens | ||
9. | ALA5205867 | 60; SJ432 | Kd | = | 6 | nM | ALA5242791 | 8.22 | nM | Homo sapiens | ||
10. | ALA5269983 | 17; SJ018 | Kd | = | 14 | nM | ALA5242791 | 7.85 | nM | Homo sapiens | ||
11. | ALA5205867 | 60; SJ432 | Kd | = | 490 | nM | ALA5242790 | 6.31 | nM | Homo sapiens | ||
12. | ALA5269983 | 17; SJ018 | Kd | = | 931 | nM | ALA5242790 | 6.03 | nM | Homo sapiens | ||
13. | ALA5274024 | 41; NEO2734 | Kd | = | 9 | nM | ALA5241955 | 8.05 | nM | Homo sapiens | ||
14. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | 7 | degrees C | ALA5236401 | degrees C | Homo sapiens | |||
15. | ALA5267793 | 9d | deltaTm | = | 1 | degrees C | ALA5236401 | degrees C | Homo sapiens | |||
16. | ALA5273240 | 34; PLX51107 | Kd | = | 5.9 | nM | ALA5232448 | 8.23 | nM | Homo sapiens | ||
17. | ALA5273240 | 34; PLX51107 | Kd | = | 1.6 | nM | ALA5232447 | 8.80 | nM | Homo sapiens | ||
18. | ALA2017287 | 34 | Kd | = | 39 | nM | ALA5232442 | 7.41 | nM | Homo sapiens | ||
19. | ALA1828978 | 1 | IC50 | = | 3 | uM | ALA5232439 | 5.52 | nM | Homo sapiens | ||
20. | ALA12543 | 18 | IC50 | = | 9 | mM | ALA5232439 | 2.05 | nM | Homo sapiens |