# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 2,6-difluoro-N-[2-fluoro-5-[5-[2-[(6-morpholin-4-ylpyridin-3-yl)amino]pyrimidin-4-yl]-2-propan-2-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamide | 26 | IC50 | = | 10 | nM | ALA1811523 | 8.00 | nM | Homo sapiens | ||
2. | ALA1866510 | SID99358600 | IC50 | = | 35.094 | uM | ALA1963838 | 4.46 | inactive | nM | Homo sapiens | |
3. | ALA1528507 | SID49644090 | IC50 | = | 3.973 | uM | ALA1963838 | 5.40 | active | nM | Homo sapiens | |
4. | ALA1438559 | SID3714531 | IC50 | = | 25.743 | uM | ALA1963838 | 4.59 | inactive | nM | Homo sapiens | |
5. | ALA1406616 | SID85146485 | IC50 | = | 11.259 | uM | ALA1963838 | 4.95 | inactive | nM | Homo sapiens | |
6. | ALA1508267 | SID24786265 | IC50 | = | 11.055 | uM | ALA1963838 | 4.96 | inactive | nM | Homo sapiens | |
7. | ALA1421321 | SID24781881 | IC50 | > | 11.957 | uM | ALA1963838 | inactive | nM | Homo sapiens | ||
8. | ALA1877372 | SID103060662 | IC50 | = | 42.901 | uM | ALA1963838 | 4.37 | inactive | nM | Homo sapiens | |
9. | ALA1975487 | SID22412240 | IC50 | = | 14.679 | uM | ALA1963838 | 4.83 | inactive | nM | Homo sapiens | |
10. | ALA1595937 | SID24802651 | IC50 | = | 9.545 | uM | ALA1963838 | 5.02 | active | nM | Homo sapiens | |
11. | ALA1729353 | SID85267991 | IC50 | > | 35.874 | uM | ALA1963838 | inactive | nM | Homo sapiens | ||
12. | ALA1345229 | SID4251053 | IC50 | = | 17.089 | uM | ALA1963838 | 4.77 | inactive | nM | Homo sapiens | |
13. | ALA1383315 | SID17506847 | IC50 | = | 4.813 | uM | ALA1963838 | 5.32 | active | nM | Homo sapiens | |
14. | ALA1709889 | SID93577001 | IC50 | = | 12.584 | uM | ALA1963838 | 4.90 | inactive | nM | Homo sapiens | |
15. | ALA1396943 | SID51086823 | IC50 | > | 35.878 | uM | ALA1963838 | inactive | nM | Homo sapiens | ||
16. | Methotrexate | 138 | IC50 | > | 35.879 | uM | ALA1963838 | inactive | nM | Homo sapiens | ||
17. | ALA1975006 | SID49644288 | IC50 | > | 11.954 | uM | ALA1963838 | inactive | nM | Homo sapiens | ||
18. | ALA1719626 | SID89855461 | IC50 | = | 8.568 | uM | ALA1963838 | 5.07 | active | nM | Homo sapiens | |
19. | ALA485636 | 14 | IC50 | > | 35.873 | uM | ALA1963838 | inactive | nM | Homo sapiens | ||
20. | ALA1373969 | SID17509718 | IC50 | = | 6.913 | uM | ALA1963838 | 5.16 | active | nM | Homo sapiens |