# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2147469 | spumigin A | EC50 | = | 0.2 | uM | ALA2148452 | 6.70 | nM | Homo sapiens | ||
2. | ALA2147467 | 1, spumigin J | EC50 | = | 0.7 | uM | ALA2148452 | 6.16 | nM | Homo sapiens | ||
3. | N-[(1R)-1-(N'-cyano-N,N'-dimethylhydrazinecarbonyl)-2-(2-methylpropanesulfonyl)ethyl]benzamide | (R)-26 | INH | 0 | ALA2156369 | tde | % | Homo sapiens | ||||
4. | N-[(1R)-1-(N'-cyano-N,N'-dimethylhydrazinecarbonyl)-2-(2-methylpropanesulfonyl)ethyl]benzamide | (R)-26 | Ki | = | 5.8 | nM | ALA2157198 | 8.24 | nM | Homo sapiens | ||
5. | ALA2153172 | (R)-22 | Ki | = | 24 | uM | ALA2157193 | 4.62 | nM | Homo sapiens | ||
6. | ALA2153171 | (+/-)-16 | Ki | = | 7.2 | uM | ALA2157193 | 5.14 | nM | Homo sapiens | ||
7. | ALA2153170 | (+/-)-15 | Ki | = | 6.8 | uM | ALA2157193 | 5.17 | nM | Homo sapiens | ||
8. | ALA2153169 | (+/-)-14 | Ki | = | 3.4 | uM | ALA2157193 | 5.47 | nM | Homo sapiens | ||
9. | ALA2153168 | (+/-)-13 | Ki | = | 3.9 | uM | ALA2157193 | 5.41 | nM | Homo sapiens | ||
10. | ALA2153167 | (+/-)-12 | Ki | = | 34 | uM | ALA2157193 | 4.47 | nM | Homo sapiens | ||
11. | ALA2153166 | (+/-)-11 | Ki | = | 5.4 | uM | ALA2157193 | 5.27 | nM | Homo sapiens | ||
12. | ALA2153165 | (+/-)-10 | Ki | = | 6.4 | uM | ALA2157193 | 5.19 | nM | Homo sapiens | ||
13. | ALA2153164 | (+/-)-9 | Ki | = | 5.1 | uM | ALA2157193 | 5.29 | nM | Homo sapiens | ||
14. | ALA2153163 | (+/-)-8 | Ki | = | 24 | uM | ALA2157193 | 4.62 | nM | Homo sapiens | ||
15. | ALA2153162 | (+/-)-7 | Ki | = | 40 | uM | ALA2157193 | 4.40 | nM | Homo sapiens | ||
16. | Cerpegin | 1, Norcerpegin | INH | 0 | ALA3128831 | Not Active | % | Homo sapiens | ||||
17. | ALA3128254 | 2 | INH | 0 | ALA3128831 | Not Active | % | Homo sapiens | ||||
18. | ALA3128255 | 3 | INH | 0 | ALA3128831 | Not Active | % | Homo sapiens | ||||
19. | ALA3128256 | 4 | INH | 0 | ALA3128831 | Not Active | % | Homo sapiens | ||||
20. | ALA3128257 | 5 | INH | 0 | ALA3128831 | Not Active | % | Homo sapiens |