| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA603656 | 29b | IC50 | = | 6 | uM | ALA3762006 | 5.22 | nM | Homo sapiens | ||
| 2. |  ALA270050 | 10a | IC50 | = | 59 | uM | ALA3762006 | 4.23 | nM | Homo sapiens | ||
| 3. |  4-{[1-Methyl-2,4-Dioxo-6-(3-Phenylprop-1-Yn-1-Yl)-1,4-Dihydroquinazolin-3(2h)-Yl]methyl}benzoic Acid | 26 | IC50 | = | 18 | uM | ALA3762006 | 4.75 | nM | Homo sapiens | ||
| 4. |  ALA5279298 | 12l | Activity | 0 | ALA5223923 | Not Active | Homo sapiens | |||||
| 5. | ALA5279298 | 12l | INH | 0 | ALA5223917 | Not Active | % | Homo sapiens | ||||
| 6. |  ALA5199698 | 58 | IC50 | > | 50 | uM | ALA5161228 | nM | Homo sapiens | |||
| 7. |  estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | FC | = | 17 | ALA3528450 | Homo sapiens | |||||
| 8. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Ratio | = | 26 | uL/min | ALA3528447 | uL/min | Homo sapiens | |||
| 9. |  Aciclovir | 13 | Ratio | = | 1 | uL/min | ALA3528447 | uL/min | Homo sapiens | |||
| 10. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Km | = | 17 | uM | ALA3528446 | nM | Homo sapiens | |||
| 11. | Aciclovir | 13 | Km | = | 772 | uM | ALA3528446 | nM | Homo sapiens | |||
| 12. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Jmax | = | 436 | pmol/min | ALA3528445 | pmol/min | Homo sapiens | |||
| 13. | Aciclovir | 13 | Jmax | = | 797 | pmol/min | ALA3528445 | pmol/min | Homo sapiens | |||
| 14. |  Penciclovir | 3 Penciclovir | Drug transport | 0 | ALA3539897 | Not Active | Homo sapiens | |||||
| 15. |  Ganciclovir | Ganciclovir | Drug transport | 0 | ALA3539894 | Not Active | Homo sapiens | |||||
| 16. | Aciclovir | 13 | FC | = | 1.7 | ALA3539892 | Homo sapiens | |||||
| 17. |  Linagliptin | 1, BI 1356 | IC50(app) | > | 100 | uM | ALA3536605 | nM | Homo sapiens | |||
| 18. |  Probenecid | probenecid | INH | = | 88.5 | % | ALA3536928 | % | Homo sapiens | |||
| 19. | Linagliptin | 1, BI 1356 | INH | = | 0 | % | ALA3536928 | % | Homo sapiens | |||
| 20. | Linagliptin | 1, BI 1356 | Drug uptake | 0 | ALA3536913 | Not Active | Homo sapiens |
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