# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | EN460 | EN460 | INH | 0 | ALA4321224 | Active | % | Homo sapiens | ||||
2. | EN460 | EN460 | IC50 | = | 22.13 | uM | ALA4321240 | 4.66 | nM | Homo sapiens | ||
3. | EN460 | EN460 | Tm | = | 55.86 | degrees C | ALA4321232 | degrees C | Homo sapiens | |||
4. | ALA4589116 | PB10 | Tm | = | 59.76 | degrees C | ALA4321232 | degrees C | Homo sapiens | |||
5. | EN460 | EN460 | INH | 0 | ALA4321230 | Dose-dependent effect | % | Homo sapiens | ||||
6. | EN460 | EN460 | IC50 | = | 12.74 | uM | ALA4321230 | 4.89 | nM | Homo sapiens | ||
7. | ALA4589116 | PB10 | INH | 0 | ALA4321230 | Dose-dependent effect | % | Homo sapiens | ||||
8. | ALA4589116 | PB10 | IC50 | = | 12.19 | uM | ALA4321230 | 4.91 | nM | Homo sapiens | ||
9. | ALA4447199 | AN968 | INH | 0 | ALA4321230 | Not Active | % | Homo sapiens | ||||
10. | ALA4528667 | Ak968 | INH | 0 | ALA4321230 | Active | % | Homo sapiens | ||||
11. | ALA1668300 | 12 | IC50 | = | 80 | uM | ALA1670746 | 4.10 | nM | Homo sapiens | ||
12. | ALA1668299 | 11 | IC50 | = | 24 | uM | ALA1670746 | 4.62 | nM | Homo sapiens | ||
13. | ALA1668298 | 10 | IC50 | = | 17 | uM | ALA1670746 | 4.77 | nM | Homo sapiens | ||
14. | ALA1668297 | 9 | IC50 | = | 11 | uM | ALA1670746 | 4.96 | nM | Homo sapiens | ||
15. | ALA1668296 | 8 | IC50 | = | 37 | uM | ALA1670746 | 4.43 | nM | Homo sapiens | ||
16. | ALA1668295 | 7 | IC50 | = | 10 | uM | ALA1670746 | 5.00 | nM | Homo sapiens | ||
17. | ALA1668294 | 6 | IC50 | = | 108 | uM | ALA1670746 | nM | Homo sapiens | |||
18. | ALA1668293 | 5 | IC50 | = | 67 | uM | ALA1670746 | 4.17 | nM | Homo sapiens | ||
19. | ALA1668292 | 4 | IC50 | = | 54 | uM | ALA1670746 | 4.27 | nM | Homo sapiens | ||
20. | ALA1668291 | 3 | IC50 | = | 8 | uM | ALA1670746 | 5.10 | nM | Homo sapiens |