# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Gymnemic acid I | 1 | Ratio | = | 1.535 | ALA4270835 | Homo sapiens | |||||
2. | TG100-115 | 6 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
3. | Dinaciclib (SCH727965) | DINACICLIB | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
4. | R547 | 39, R547 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
5. | PX-866 | 4, PX-866 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
6. | AMG-900 | SID137275938 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
7. | Cobimetinib | 1, XL518, GDC-0973 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
8. | ALA1822792 | MK-2461 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
9. | ALA1614701 | AZD-6244 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
10. | Binimetinib | SID174006430 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
11. | Lapatinib | GW-572016 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
12. | Ruxolitinib (INCB018424) | 3, INCB-018424 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
13. | JNJ-38877605 | SID137276033 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
14. | ALA3545137 | PF-00477736 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
15. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
16. | ALA91829 | 1 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
17. | Sunitinib | 12b | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
18. | PF-04217903 | SID103905666 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
19. | CO-1686 (AVL-301) | ROCILETINIB | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens | ||
20. | racemic-tofacitinib | CP-690550 | Kd apparent | > | 30000 | nM | ALA3991866 | Inactive | nM | Homo sapiens |