| # | Name | Compound Key | Action Type | Relation | Activety Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4637208 | EUB0001113 | pKd | 5.1 | ALA4886881 | nM | Homo sapiens | |||||
| 2. |  ALA4639128 | 62 | Kd | 30000 | nM | ALA4886826 | nM | Homo sapiens | ||||
| 3. |  GSK620 | 1; 20 | pKd | 4.5 | ALA4885823 | nM | Homo sapiens | |||||
| 4. |  GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885763 | nM | Homo sapiens | ||||
| 5. |  ALA4648362 | EUB0001116 | pKd | 4.5 | ALA4885699 | nM | Homo sapiens | |||||
| 6. |  BAZ2-ICR | 13, BAZ2-ICR | deltaTm | = | 3.8 | degrees C | ALA3419229 | degrees C | Homo sapiens | |||
| 7. | BAZ2-ICR | 13, BAZ2-ICR | Kd | = | 170 | nM | ALA3419227 | 6.77 | nM | Homo sapiens | ||
| 8. | BAZ2-ICR | 13, BAZ2-ICR | IC50 | = | 0.18 | uM | ALA3419225 | 6.75 | nM | Homo sapiens | ||
| 9. |  ALA3415186 | 12 | IC50 | = | 2.45 | uM | ALA3419225 | 5.61 | nM | Homo sapiens | ||
| 10. |  ALA3415185 | 11 | IC50 | = | 0.79 | uM | ALA3419225 | 6.10 | nM | Homo sapiens | ||
| 11. |  ALA3415184 | 10 | IC50 | = | 0.77 | uM | ALA3419225 | 6.11 | nM | Homo sapiens | ||
| 12. |  ALA3415183 | 8 | IC50 | > | 50 | uM | ALA3419225 | nM | Homo sapiens | |||
| 13. |  4-[5-(1-methylpyrazol-4-yl)-3-[2-(4-methyltriazol-1-yl)ethyl]imidazol-4-yl]benzonitrile | 7 | IC50 | = | 1.07 | uM | ALA3419225 | 5.97 | nM | Homo sapiens | ||
| 14. |  ALA3415181 | 6 | IC50 | > | 50 | uM | ALA3419225 | nM | Homo sapiens | |||
| 15. |  ALA3415180 | 5 | IC50 | > | 50 | uM | ALA3419225 | nM | Homo sapiens | |||
| 16. |  ALA3415179 | 4 | IC50 | = | 5.25 | uM | ALA3419225 | 5.28 | nM | Homo sapiens | ||
| 17. |  4-[3-[2-(4-methyltriazol-1-yl)ethyl]-5-phenylimidazol-4-yl]benzonitrile | 1 | IC50 | = | 26 | uM | ALA3419225 | 4.58 | nM | Homo sapiens | ||
| 18. |  ALA3415177 | 2 | IC50 | = | 4.4 | uM | ALA3419225 | 5.36 | nM | Homo sapiens | ||
| 19. |  ALA3415178 | 3 | IC50 | > | 50 | uM | ALA3419225 | nM | Homo sapiens | |||
| 20. |  GSK1324726A (I-BET726) | 45 | pIC50 | < | 4.5 | ALA3383406 | nM | Homo sapiens |
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