| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | -1 | degrees C | ALA5236406 | degrees C | Homo sapiens | |||
| 2. |  ALA5267793 | 9d | deltaTm | = | -2 | degrees C | ALA5236406 | degrees C | Homo sapiens | |||
| 3. |  GSK 4027 | (R,R)-32; GSK4027 | Ki | = | 840 | nM | ALA5214219 | 6.08 | nM | Homo sapiens | ||
| 4. |  GSK 2801 | 1 | Kd | = | 136 | nM | ALA5214169 | 6.87 | nM | Homo sapiens | ||
| 5. | GSK 2801 | 1 | dTm | = | 2.7 | K | ALA5214168 | K | Homo sapiens | |||
| 6. | GSK 2801 | 1 | Kd | = | 0.1 | uM | ALA5214167 | 7.00 | nM | Homo sapiens | ||
| 7. |  BAZ2-ICR | 13, BAZ2-ICR | dTm | = | 3.8 | K | ALA5214129 | K | Homo sapiens | |||
| 8. | GSK 2801 | 1 | IC50 | = | 430 | nM | ALA5210539 | 6.37 | nM | Homo sapiens | ||
| 9. | BAZ2-ICR | 13, BAZ2-ICR | Kd | = | 170 | nM | ALA5210531 | 6.77 | nM | Homo sapiens | ||
| 10. |  GSK8573 | 23; GSK8573 | Kd | > | 10000 | nM | ALA5210251 | nM | Homo sapiens | |||
| 11. | GSK 2801 | 1 | Kd | = | 3162 | nM | ALA5210242 | 5.50 | nM | Homo sapiens | ||
| 12. | BAZ2-ICR | 13, BAZ2-ICR | EC50 | < | 1000 | nM | ALA5210235 | nM | Homo sapiens | |||
| 13. | GSK8573 | 23; GSK8573 | IC50 | > | 100000 | nM | ALA5210069 | nM | Homo sapiens | |||
| 14. | GSK 2801 | 1 | IC50 | < | 1000 | nM | ALA5210067 | nM | Homo sapiens | |||
| 15. |  ALA5204783 | 8m | deltaTm | = | -1 | degrees C | ALA5162520 | degrees C | Homo sapiens | |||
| 16. |  ALA5206088 | 8l; XY153 | deltaTm | = | -0.25 | degrees C | ALA5162520 | degrees C | Homo sapiens | |||
| 17. |  ALA5205742 | 8k | deltaTm | = | -1 | degrees C | ALA5162520 | degrees C | Homo sapiens | |||
| 18. |  ALA5178480 | 8j | deltaTm | = | -0.75 | degrees C | ALA5162520 | degrees C | Homo sapiens | |||
| 19. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | -0.5 | degrees C | ALA5162520 | degrees C | Homo sapiens | |||
| 20. |  ALA5179520 | 9g; Y08284 | deltaTm | = | 0 | degrees C | ALA5156574 | degrees C | Homo sapiens |
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