| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Km | = | 16.1 | uM | ALA3538499 | nM | Homo sapiens | |||
| 2. |  [³H]taurocholic acid | THCA | Km | = | 15.9 | uM | ALA3538499 | nM | Homo sapiens | |||
| 3. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Vmax | = | 39.4 | pmol/mg/min | ALA3538499 | pmol/mg/min | Homo sapiens | |||
| 4. | [³H]taurocholic acid | THCA | Vmax | = | 24.1 | pmol/mg/min | ALA3538499 | pmol/mg/min | Homo sapiens | |||
| 5. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Km | = | 9.6 | uM | ALA3538512 | nM | Homo sapiens | |||
| 6. |  5-Aminosalicylic acid | 5-ASA | INH | 0 | ALA3540645 | Dose-dependent effect | % | Homo sapiens | ||||
| 7. |  ALA4645514 | 1 | Activity | 0 | ALA4624656 | Active | Homo sapiens | |||||
| 8. | ALA4645514 | 1 | Activity | 0 | ALA4624657 | Not Active | Homo sapiens | |||||
| 9. |  ALA294616 | DPDPE | Activity | 0 | ALA2076566 | inhibitor [(at a rough estimate) 50 % of control] | Homo sapiens | |||||
| 10. |  DAMGO TFA | DAMGO | Activity | 0 | ALA2076567 | inhibitor [(at a rough estimate) 50 % of control] | Homo sapiens | |||||
| 11. |  ALA8234 | Leu-enkephaline | Activity | 0 | ALA2076564 | inhibitor [(at a rough estimate) 40 % of control] | Homo sapiens | |||||
| 12. |  Rifampicin | rifampacin | Ki | = | 51 | uM | ALA2076348 | 4.29 | inhibitor [Ki=51uM] | nM | Homo sapiens | |
| 13. |  Naloxone | naloxone | Activity | 0 | ALA2076563 | inhibitor [(at a rough estimate) 20 % of control] | Homo sapiens | |||||
| 14. |  ALA4297251 | Orange juice | Activity | 0 | ALA2076557 | inhibitor [(at a rough estimate) 10 % of control] | Homo sapiens | |||||
| 15. |  ALA2074618 | Grapefruit juice | Activity | 0 | ALA2076558 | inhibitor [(at a rough estimate) 10 % of control] | Homo sapiens | |||||
| 16. |  ALA567175 | 1, NTI | Activity | 0 | ALA2076562 | inhibitor [(at a rough estimate) 10 % of control] | Homo sapiens | |||||
| 17. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Activity | 0 | ALA2076565 | inhibitor [(at a rough estimate) 10 % of control] | Homo sapiens | |||||
| 18. |  Unoprostone isopropyl ester | UNOPROSTONE ISOPROPYL | Activity | 0 | ALA2076346 | is not a substrate [(-)] | Homo sapiens | |||||
| 19. |  Glycyrrhizic acid | GL (glycyrrhizin) | Activity | 0 | ALA2076561 | is not an inhibitor [-] | Homo sapiens | |||||
| 20. | Rifampicin | rifampacin | Activity | 0 | ALA2075957 | is not a substrate [-] | Homo sapiens |
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