# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA294616 | DPDPE | Activity | 0 | ALA2076566 | inhibitor [(at a rough estimate) 50 % of control] | Homo sapiens | |||||
2. | DAMGO TFA | DAMGO | Activity | 0 | ALA2076567 | inhibitor [(at a rough estimate) 50 % of control] | Homo sapiens | |||||
3. | ALA8234 | Leu-enkephaline | Activity | 0 | ALA2076564 | inhibitor [(at a rough estimate) 40 % of control] | Homo sapiens | |||||
4. | Rifampicin | rifampacin | Ki | = | 51 | uM | ALA2076348 | 4.29 | inhibitor [Ki=51uM] | nM | Homo sapiens | |
5. | [³H]naloxone | naloxone | Activity | 0 | ALA2076563 | inhibitor [(at a rough estimate) 20 % of control] | Homo sapiens | |||||
6. | ALA4297251 | Orange juice | Activity | 0 | ALA2076557 | inhibitor [(at a rough estimate) 10 % of control] | Homo sapiens | |||||
7. | ALA2074618 | Grapefruit juice | Activity | 0 | ALA2076558 | inhibitor [(at a rough estimate) 10 % of control] | Homo sapiens | |||||
8. | ALA567175 | 1, NTI | Activity | 0 | ALA2076562 | inhibitor [(at a rough estimate) 10 % of control] | Homo sapiens | |||||
9. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | Activity | 0 | ALA2076565 | inhibitor [(at a rough estimate) 10 % of control] | Homo sapiens | |||||
10. | Unoprostone isopropyl ester | UNOPROSTONE ISOPROPYL | Activity | 0 | ALA2076346 | is not a substrate [(-)] | Homo sapiens | |||||
11. | Glycyrrhizic acid | GL (glycyrrhizin) | Activity | 0 | ALA2076561 | is not an inhibitor [-] | Homo sapiens | |||||
12. | Rifampicin | rifampacin | Activity | 0 | ALA2075957 | is not a substrate [-] | Homo sapiens | |||||
13. | Enalapril | 2 | Activity | 0 | ALA2075958 | is not a substrate [-] | Homo sapiens | |||||
14. | Pravastatin | 2 (pravastatin) | Activity | 0 | ALA2076111 | is not a substrate [-] | Homo sapiens | |||||
15. | rifamycin SV | 1b(rifamycin SV) | Ki | = | 11 | uM | ALA2076348 | 4.96 | inhibitor [Ki=11uM] | nM | Homo sapiens | |
16. | Unoprostone | unoprostone | Km | = | 93 | uM | ALA2076346 | substrate [Km=93uM] | nM | Homo sapiens | ||
17. | [³H]taurocholic acid | THCA | Km | = | 93 | uM | ALA2077847 | substrate [Km=93uM] | nM | Homo sapiens | ||
18. | L-Thyroxine | 181 (Thyroxine) | Km | = | 8 | uM | ALA2077861 | substrate [Km=8uM] | nM | Homo sapiens | ||
19. | [³H]taurocholic acid | THCA | Km | = | 64 | uM | ALA2076112 | substrate [Km=64uM] | nM | Homo sapiens | ||
20. | [³H]taurocholic acid | THCA | Km | = | 60 | uM | ALA2077847 | substrate [Km=60uM] | nM | Homo sapiens |