# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Oseltamivir | oseltamivir | Drug uptake | 0 | ALA3536471 | Not Active | Homo sapiens | |||||
2. | Oseltamivir Acid | 1 (GS-4071) | Drug uptake | 0 | ALA3536471 | Not Active | Homo sapiens | |||||
3. | L-Carnosine | Carnosine (beta-ala his) | EC50 | = | 28 | uM | ALA5209612 | 4.55 | Substrate; At Ph 6.8 | nM | Homo sapiens | |
4. | glycyl-sarcosine | 38 | EC50 | = | 39 | uM | ALA5209612 | 4.41 | Substrate; At Ph 6.8 | nM | Homo sapiens | |
5. | glycyl-sarcosine | 38 | EC50 | = | 123 | uM | ALA5209612 | Substrate; At Ph 7.4 | nM | Homo sapiens | ||
6. | ALA66839 | 7/ DK | Ki | = | 8 | uM | ALA2077099 | 5.10 | inhibitor [Ki=8uM] | nM | Homo sapiens | |
7. | Ala-Ala | 10 | Ki | = | 6 | uM | ALA2077099 | 5.22 | inhibitor [Ki=6uM] | nM | Homo sapiens | |
8. | Cephalexin | 5 | Ki | = | 68.2 | uM | ALA2076904 | 4.17 | inhibitor [Ki=68.2uM] | nM | Homo sapiens | |
9. | glycyl-sarcosine | 38 | Ki | = | 64 | uM | ALA2077645 | 4.19 | inhibitor [Ki=64uM] | nM | Homo sapiens | |
10. | cyclacillin | 83(Cyclacillin) | Ki | = | 39.1 | uM | ALA2076904 | 4.41 | inhibitor [Ki=39.1uM] | nM | Homo sapiens | |
11. | cyclacillin | 83(Cyclacillin) | Ki | = | 36.8 | uM | ALA2075812 | 4.43 | inhibitor [Ki=36.8uM] | nM | Homo sapiens | |
12. | ALA93178 | KA | Ki | = | 23 | uM | ALA2077099 | 4.64 | inhibitor [Ki=23uM] | nM | Homo sapiens | |
13. | Cefadroxil | 85(Cefadroxil) | Ki | = | 2.8 | uM | ALA2076904 | 5.55 | inhibitor [Ki=2.8uM] | nM | Homo sapiens | |
14. | Cefadroxil | 85(Cefadroxil) | Ki | = | 2.5 | uM | ALA2075812 | 5.60 | inhibitor [Ki=2.5uM] | nM | Homo sapiens | |
15. | ALA380047 | 91 | Ki | = | 18 | uM | ALA2077099 | 4.75 | inhibitor [Ki=18uM] | nM | Homo sapiens | |
16. | ALA191057 | 115 | Ki | = | 11 | uM | ALA2077099 | 4.96 | inhibitor [Ki=11uM] | nM | Homo sapiens | |
17. | Cefadroxil | 85(Cefadroxil) | IC50 | = | 66 | uM | ALA2075813 | 4.18 | inhibitor [IC50=66uM] | nM | Homo sapiens | |
18. | cyclacillin | 83(Cyclacillin) | IC50 | = | 610 | uM | ALA2075813 | inhibitor [IC50=610uM] | nM | Homo sapiens | ||
19. | glycyl-sarcosine | 38 | Km | = | 74 | uM | ALA2077646 | substrate [Km=74uM] | nM | Homo sapiens | ||
20. | glycyl-sarcosine | 38 | Km | = | 48 | uM | ALA2077644 | substrate [Km=48uM] | nM | Homo sapiens |