# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | IC50 | = | 95 | uM | ALA2077067 | 4.02 | inhibitor [IC50=95uM] | nM | Homo sapiens | |
2. | ALA2074982 | Dehydroepiandrosterone-3-glucuronide | IC50 | = | 80 | uM | ALA2077531 | 4.10 | inhibitor [IC50=80uM] | nM | Homo sapiens | |
3. | ALA2074982 | Dehydroepiandrosterone-3-glucuronide | IC50 | = | 80 | uM | ALA2077067 | 4.10 | inhibitor [IC50=80uM] | nM | Homo sapiens | |
4. | ALA2074591 | Estradiol-3-glucuronide | IC50 | = | 80 | uM | ALA2077067 | 4.10 | inhibitor [IC50=80uM] | nM | Homo sapiens | |
5. | S-(4-Nitrobenzyl)-6-thioinosine | 6n | IC50 | = | 75 | uM | ALA2077068 | 4.12 | inhibitor [IC50=75uM] | nM | Homo sapiens | |
6. | ALA3349339 | Estradiol 3-sulfate | IC50 | = | 70 | uM | ALA2077067 | 4.16 | inhibitor [IC50=70uM] | nM | Homo sapiens | |
7. | Taurodeoxychloic acid | 7a, tauro | IC50 | = | 60 | uM | ALA2078156 | 4.22 | inhibitor [IC50=60uM] | nM | Homo sapiens | |
8. | Taurochenodeoxycholic acid | 7 | IC50 | = | 55 | uM | ALA2078156 | 4.26 | inhibitor [IC50=55uM] | nM | Homo sapiens | |
9. | ALA3349339 | Estradiol 3-sulfate | IC50 | = | 50 | uM | ALA2077531 | 4.30 | inhibitor [IC50=50uM] | nM | Homo sapiens | |
10. | estrone-3-sulphate | estrone-3-O-sulfamate (EMATE) | IC50 | = | 45 | uM | ALA2077531 | 4.35 | inhibitor [IC50=45uM] | nM | Homo sapiens | |
11. | Glycocholic acid | 5b, glyco | IC50 | = | 400 | uM | ALA2078156 | inhibitor [IC50=400uM] | nM | Homo sapiens | ||
12. | Dehydroepiandrosterone sulfate | Dehydroepiandrosterone sulfate (DHEAS) | IC50 | = | 3 | uM | ALA2078640 | 5.52 | inhibitor [IC50=3uM] | nM | Homo sapiens | |
13. | [³H]taurocholic acid | THCA | IC50 | = | 350 | uM | ALA2078156 | inhibitor [IC50=350uM] | nM | Homo sapiens | ||
14. | [³H]estradiol-17β-glucuronide | estradiol 17b glucuronide | IC50 | = | 30 | uM | ALA2077067 | 4.52 | inhibitor [IC50=30uM] | nM | Homo sapiens | |
15. | estradiol disulfate | estradiol disulfate | IC50 | = | 2 | uM | ALA2077531 | 5.70 | inhibitor [IC50=2uM] | nM | Homo sapiens | |
16. | Dipyridamole | Dipyridamole | IC50 | = | 2 | uM | ALA2077068 | 5.70 | inhibitor [IC50=2uM] | nM | Homo sapiens | |
17. | [³H]taurocholic acid | THCA | IC50 | = | 250 | uM | ALA2078641 | inhibitor [IC50=250uM] | nM | Homo sapiens | ||
18. | taurolithocholic acid-3-sulphate | 6a, tauro | IC50 | = | 20 | uM | ALA2078156 | 4.70 | inhibitor [IC50=20uM] | nM | Homo sapiens | |
19. | dilazep | Dilazep | IC50 | = | 20 | uM | ALA2077068 | 4.70 | inhibitor [IC50=20uM] | nM | Homo sapiens | |
20. | Sildenafil | 1 | IC50 | = | 20 | uM | ALA2077068 | 4.70 | inhibitor [IC50=20uM] | nM | Homo sapiens |