| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1402 | 3 | Km(app) | = | 2.6 | uM | ALA3540601 | nM | Homo sapiens | |||
| 2. | ALA1402 | 3 | Vmax | = | 8.5 | nmol/min | ALA3540604 | nmol/min | Homo sapiens | |||
| 3. |  β-Estradiol | Table II | Km | = | 2.4 | uM | ALA3537867 | nM | Homo sapiens | |||
| 4. | β-Estradiol | Table II | Vmax | = | 16 | pmol/min/ug | ALA3537867 | pmol/min/ug | Homo sapiens | |||
| 5. | β-Estradiol | Table II | Km | = | 0.36 | uM | ALA3537868 | nM | Homo sapiens | |||
| 6. |  Ethinyl Estradiol | 17 alpha-ethynyl E2 | Km | = | 0.69 | uM | ALA3537869 | nM | Homo sapiens | |||
| 7. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | Vmax | = | 11 | pmol/min/ug | ALA3537869 | pmol/min/ug | Homo sapiens | |||
| 8. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | Km | = | 0.45 | uM | ALA3537870 | nM | Homo sapiens | |||
| 9. | β-Estradiol | Table II | Kd | = | 2.3 | uM | ALA3537871 | 5.64 | nM | Homo sapiens | ||
| 10. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | Kd | = | 0.5 | uM | ALA3537871 | 6.30 | nM | Homo sapiens | ||
| 11. | β-Estradiol | Table II | Kd | = | 1.2 | uM | ALA3537872 | 5.92 | nM | Homo sapiens | ||
| 12. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | Kd | = | 4.3 | nM | ALA3537872 | 8.37 | nM | Homo sapiens | ||
| 13. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | Ki | = | 14.9 | nM | ALA3537873 | 7.83 | nM | Homo sapiens | ||
| 14. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | Ki | = | 8.9 | nM | ALA3537874 | 8.05 | nM | Homo sapiens | ||
| 15. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | Ki | = | 19 | nM | ALA3537875 | 7.72 | nM | Homo sapiens | ||
| 16. | Ethinyl Estradiol | 17 alpha-ethynyl E2 | IC50 | = | 20 | nM | ALA3537876 | 7.70 | nM | Homo sapiens | ||
| 17. |  ALA3527569 | M25 | Drug metabolism | 0 | ALA3539757 | metabolite_detected | Homo sapiens | |||||
| 18. |  Brivanib (BMS-540215) | 12 | Drug metabolism | 0 | ALA3539752 | metabolite_detected | Homo sapiens | |||||
| 19. |  2-(4-(Methylamino)phenyl)benzo[d]thiazol-6-ol | 6-Substituted BTA analogue | Ki | = | 5.1 | nM | ALA4482682 | 8.29 | nM | Homo sapiens | ||
| 20. |  ALA4557856 | 17 | Ki | = | 24 | nM | ALA4482682 | 7.62 | nM | Homo sapiens |
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