# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA301982 | 1 | Ki | = | 0.49 | uM | ALA5233905 | 6.31 | nM | Homo sapiens | ||
2. | ALA4785914 | 19 | IC50 | > | 10 | uM | ALA4731222 | nM | Homo sapiens | |||
3. | PT-2385 | (S)-10i | Drug metabolism | 0 | ALA4312546 | Metabolite_Notdetected | Homo sapiens | |||||
4. | PF-05221304 | 38 | IC50 | > | 20 | uM | ALA4669901 | nM | Homo sapiens | |||
5. | ALA3398252 | 2 | Drug metabolism | 0 | ALA3398974 | metabolite_notdetected | Homo sapiens | |||||
6. | Raltegravir (MK-0518) | 1, raltegravir | Drug metabolism | 0 | ALA3398974 | metabolite_detected | Homo sapiens | |||||
7. | ALA3398252 | 2 | Activity | 0 | ALA3398979 | Not Active | Homo sapiens | |||||
8. | ALA3398252 | 2 | IC50 | > | 300 | uM | ALA3399065 | nM | Homo sapiens | |||
9. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Drug metabolism | 0 | ALA3531820 | metabolite_detected | Homo sapiens | |||||
10. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Drug metabolism | 0 | ALA3541445 | metabolite_detected | Homo sapiens | |||||
11. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Km | = | 777.7 | uM | ALA3531836 | nM | Homo sapiens | |||
12. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Vmax | = | 1244 | pmol/min/g | ALA3531837 | pmol/min/g | Homo sapiens | |||
13. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | CL | = | 1.6 | uL/min/g | ALA3531838 | mL.min-1.g-1 | Homo sapiens | |||
14. | ALA3527359 | YM150 monomaleate | Drug metabolism | < | 0.01 | nmol/min | ALA3534355 | nmol/min | Homo sapiens | |||
15. | Dolutegravir (GSK1349572) | DOLUTEGRAVIR | Drug metabolism | 0 | ALA3541849 | metabolite_not_detected | Homo sapiens | |||||
16. | Haloperidol | Haloperidol | Drug metabolism | 0 | ALA3539919 | metabolite_not_detected | Homo sapiens | |||||
17. | Haloperidol | Haloperidol | Drug metabolism | 0 | ALA3539909 | metabolite_not_detected | Homo sapiens | |||||
18. | ALA3527027 | Lorcaserin | Drug metabolism | 0 | ALA3534328 | metabolite_detected | Homo sapiens | |||||
19. | ALA3527103 | [14C]-Rivoglitazone | Drug metabolism | 0 | ALA3541112 | metabolite_not_detected | Homo sapiens | |||||
20. | ALA3527103 | [14C]-Rivoglitazone | Drug metabolism | 0 | ALA3529365 | metabolite_not_detected | Homo sapiens |