# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PT-2385 | (S)-10i | Drug metabolism | 0 | ALA4312547 | Metabolite_Notdetected | Homo sapiens | |||||
2. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Drug metabolism | 0 | ALA3531818 | metabolite_detected | Homo sapiens | |||||
3. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Drug metabolism | 0 | ALA3541446 | metabolite_detected | Homo sapiens | |||||
4. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Km | = | 432.3 | uM | ALA3531839 | nM | Homo sapiens | |||
5. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Vmax | = | 740.2 | pmol/min/g | ALA3531840 | pmol/min/g | Homo sapiens | |||
6. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | CL | = | 1.7 | uL/min/g | ALA3531841 | mL.min-1.g-1 | Homo sapiens | |||
7. | ALA3527359 | YM150 monomaleate | CL | = | 12.3 | uL/min/g | ALA3534362 | mL.min-1.g-1 | Homo sapiens | |||
8. | ALA3527359 | YM150 monomaleate | Vmax | = | 0.725 | nmol/min | ALA3534361 | nmol/min | Homo sapiens | |||
9. | ALA3527359 | YM150 monomaleate | Km | = | 59.1 | uM | ALA3534360 | nM | Homo sapiens | |||
10. | ALA3527359 | YM150 monomaleate | Drug metabolism | = | 0.251 | nmol/min | ALA3534351 | nmol/min | Homo sapiens | |||
11. | Haloperidol | Haloperidol | Drug metabolism | 0 | ALA3539920 | metabolite_not_detected | Homo sapiens | |||||
12. | Haloperidol | Haloperidol | Drug metabolism | 0 | ALA3539910 | metabolite_not_detected | Homo sapiens | |||||
13. | 16-Epiestriol | 16-Epiestriol | Drug metabolism | = | 0.5 | pmol/min/mg | ALA3532971 | pmol/min/mg | Homo sapiens | |||
14. | ALA3527103 | [14C]-Rivoglitazone | Drug metabolism | 0 | ALA3541114 | metabolite_not_detected | Homo sapiens | |||||
15. | ALA3527103 | [14C]-Rivoglitazone | Drug metabolism | 0 | ALA3529366 | metabolite_not_detected | Homo sapiens | |||||
16. | ALA3527103 | [14C]-Rivoglitazone | Drug metabolism | 0 | ALA3530954 | metabolite_not_detected | Homo sapiens | |||||
17. | ALA3527579 | 3'-OH-TCC | Drug metabolism | = | 1700 | pmol/min/mg | ALA3534071 | pmol/min/mg | Homo sapiens | |||
18. | ALA3527500 | 2'-OH-TCC | Drug metabolism | = | 870 | pmol/min/mg | ALA3534071 | pmol/min/mg | Homo sapiens | |||
19. | AMG 853 | 5, AMG-853 | Drug metabolism | 0 | ALA3528028 | metabolite_not_detected | Homo sapiens | |||||
20. | 3,4,4'-Trichlorocarbanilide | 16 | Drug metabolism | 0 | ALA3538804 | metabolite_not_detected | Homo sapiens |