# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4442951 | DHD3; D2 | Activity | = | 45 | % | ALA4378686 | % | Homo sapiens | |||
2. | ALA4550375 | DHD1; D1 | Activity | = | 12 | % | ALA4378686 | % | Homo sapiens | |||
3. | ALA4452336 | 8 | t1/2 | = | 11 | min | ALA4339116 | hr | Homo sapiens | |||
4. | ALA4483087 | 7 | t1/2 | = | 2.9 | min | ALA4339116 | hr | Homo sapiens | |||
5. | Epacadostat (INCB024360) | EPACADOSTAT | t1/2 | = | 23 | min | ALA4339116 | hr | Homo sapiens | |||
6. | ALA4449948 | 28 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
7. | ALA4475499 | 27 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
8. | ALA4461796 | 26 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
9. | ALA4441030 | 25 | t1/2 | = | 57.3 | min | ALA4339116 | hr | Homo sapiens | |||
10. | ALA4585089 | 24 | t1/2 | = | 54 | min | ALA4339116 | hr | Homo sapiens | |||
11. | ALA4465837 | 23 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
12. | ALA4439896 | 22 | t1/2 | = | 86.7 | min | ALA4339116 | hr | Homo sapiens | |||
13. | ALA4533432 | 21 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
14. | ALA4437616 | 20 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
15. | ALA4538516 | 19 | t1/2 | = | 104 | min | ALA4339116 | hr | Homo sapiens | |||
16. | ALA4521926 | 18 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
17. | ALA4549976 | 17 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
18. | ALA4441246 | 16 | t1/2 | = | 95.2 | min | ALA4339116 | hr | Homo sapiens | |||
19. | ALA4455438 | 15 | t1/2 | > | 180 | min | ALA4339116 | hr | Homo sapiens | |||
20. | ALA4578545 | 14 | t1/2 | = | 91.8 | min | ALA4339116 | hr | Homo sapiens |