| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3527060 | M6 | kobs | = | 0.42 | /min | ALA3535629 | /min | Oryctolagus cuniculus | |||
| 2. |  Ticlopidine | Ticlopidine | Compound recovery | 0 | ALA3538996 | metabolite_detected | Oryctolagus cuniculus | |||||
| 3. | Ticlopidine | Ticlopidine | Compound recovery | 0 | ALA3538995 | metabolite_detected | Oryctolagus cuniculus | |||||
| 4. |  ALA3526247 | M3 | Compound recovery | 0 | ALA3538999 | metabolite_detected | Oryctolagus cuniculus | |||||
| 5. |  ALA3526245 | M1 | Compound recovery | 0 | ALA3538999 | metabolite_detected | Oryctolagus cuniculus | |||||
| 6. | Ticlopidine | Ticlopidine | Compound recovery | 0 | ALA3538994 | metabolite_detected | Oryctolagus cuniculus | |||||
| 7. | Ticlopidine | Ticlopidine | Compound recovery | 0 | ALA3541181 | metabolite_detected | Oryctolagus cuniculus | |||||
| 8. | Ticlopidine | Ticlopidine | Compound recovery | 0 | ALA3538997 | metabolite_detected | Oryctolagus cuniculus | |||||
| 9. |  ALA3526246 | M2 | Compound recovery | 0 | ALA3538999 | metabolite_detected | Oryctolagus cuniculus | |||||
| 10. |  ALA3526248 | M4 | Compound recovery | 0 | ALA3538999 | metabolite_detected | Oryctolagus cuniculus | |||||
| 11. |  Ticlopidine N-Oxide | M5 | Compound recovery | 0 | ALA3538999 | metabolite_detected | Oryctolagus cuniculus | |||||
| 12. | ALA3526245 | M1 | kobs | = | 0.49 | /min | ALA3535629 | /min | Oryctolagus cuniculus | |||
| 13. | ALA3526246 | M2 | kobs | = | 0.48 | /min | ALA3535629 | /min | Oryctolagus cuniculus | |||
| 14. | ALA3526248 | M4 | kobs | = | 0.56 | /min | ALA3535629 | /min | Oryctolagus cuniculus | |||
| 15. | Ticlopidine N-Oxide | M5 | kobs | = | 0.66 | /min | ALA3535629 | /min | Oryctolagus cuniculus | |||
| 16. | Ticlopidine | Ticlopidine | Kinact | = | 0.5 | /min | ALA3535631 | /min | Oryctolagus cuniculus | |||
| 17. |  bupropion | bupropion | Kinact | = | 0.08 | /min | ALA3535631 | /min | Oryctolagus cuniculus | |||
| 18. |  ALA3527032 | 7-EFC | Kinact | = | 0.02 | /min | ALA3535631 | /min | Oryctolagus cuniculus | |||
| 19. |  Bergamottin | 4 | Kinact | = | 0.068 | min-1 | ALA1743487 | Cytochrome P450 mechanistic inhibitor: PMID 15608076 | min-1 | Oryctolagus cuniculus | ||
| 20. | Bergamottin | 4 | KI | = | 2.8 | uM | ALA1743487 | 5.55 | Cytochrome P450 mechanistic inhibitor: PMID 15608076 | nM | Oryctolagus cuniculus |
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