| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3526300 | [3H]Tiotropium | Drug uptake | 0 | ALA3531417 | Not Active | Rattus norvegicus | |||||
| 2. |  ALA1201053 | [3H]Ipratropium | FC | = | 5.1 | ALA3531417 | Rattus norvegicus | |||||
| 3. |  PF-04971729 | 4, PF-04971729 | INH | 0 | ALA1771938 | Not Active | % | Rattus norvegicus | ||||
| 4. |  Corticosterone | 7 | Activity | 0 | ALA2078042 | inhibitor [(at a rough estimate) 5 % of control] | Rattus norvegicus | |||||
| 5. |  5-Hydroxytryptamine | 1a | IC50 | = | 97 | uM | ALA2077839 | 4.01 | inhibitor [IC50=97uM] | nM | Rattus norvegicus | |
| 6. |  11-Deoxy Corticosterone | table VI | IC50 | = | 8.4 | uM | ALA2077061 | 5.08 | inhibitor [IC50=8.4uM] | nM | Rattus norvegicus | |
| 7. |  desipramine | desmethylimipramine | IC50 | = | 68 | uM | ALA2077839 | 4.17 | inhibitor [IC50=68uM] | nM | Rattus norvegicus | |
| 8. |  4-(2-Aminoethyl)benzene-1,2-diol | Dopamine | IC50 | = | 62 | uM | ALA2077839 | 4.21 | inhibitor [IC50=62uM] | nM | Rattus norvegicus | |
| 9. |  L-Noradrenaline | NE | IC50 | = | 434 | uM | ALA2077061 | inhibitor [IC50=434uM] | nM | Rattus norvegicus | ||
| 10. |  amphetamine | 4 (+/-) | IC50 | = | 42 | uM | ALA2077839 | 4.38 | inhibitor [IC50=42uM] | nM | Rattus norvegicus | |
| 11. | Corticosterone | 7 | IC50 | = | 4.9 | uM | ALA2077061 | 5.31 | inhibitor [IC50=4.9uM] | nM | Rattus norvegicus | |
| 12. | 4-(2-Aminoethyl)benzene-1,2-diol | Dopamine | IC50 | = | 384 | uM | ALA2077061 | inhibitor [IC50=384uM] | nM | Rattus norvegicus | ||
| 13. |  ALA1201201 | 5 | IC50 | = | 248 | uM | ALA2077839 | inhibitor [IC50=248uM] | nM | Rattus norvegicus | ||
| 14. |  MPP⁺ | 1 | Km | = | 91 | uM | ALA2075859 | substrate [Km=91uM] | nM | Rattus norvegicus | ||
| 15. |  ALA103 | Progesterone | IC50 | = | 10.5 | uM | ALA2077061 | 4.98 | inhibitor [IC50=10.5uM] | nM | Rattus norvegicus | |
| 16. |  β-Estradiol | Table II | IC50 | = | 1.1 | uM | ALA2077061 | 5.96 | inhibitor [IC50=1.1uM] | nM | Rattus norvegicus | |
| 17. |  agmatine | Agmatine | Km | = | 900 | uM | ALA2075860 | substrate [Km=900uM] | nM | Rattus norvegicus | ||
| 18. |  tetraethylammonium | 1 | Km | = | 6200 | uM | ALA2078030 | substrate [Km=6200uM] | nM | Rattus norvegicus | ||
| 19. | tetraethylammonium | 1 | Km | = | 2500 | uM | ALA2075858 | substrate [Km=2500uM] | nM | Rattus norvegicus | ||
| 20. | MPP⁺ | 1 | Km | = | 24 | uM | ALA2078029 | substrate [Km=24uM] | nM | Rattus norvegicus |
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