| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  PF 04991532 | 19 | Drug uptake | 0 | ALA2166281 | Not Active | Rattus norvegicus | |||||
| 2. |  Probenecid | probenecid | Ki | = | 72.9 | uM | ALA2077473 | 4.14 | inhibitor [Ki=72.9uM] | nM | Rattus norvegicus | |
| 3. |  rifamycin SV | 1b(rifamycin SV) | Ki | = | 7.3 | uM | ALA2075975 | 5.14 | inhibitor [Ki=7.3uM] | nM | Rattus norvegicus | |
| 4. |  [³H]taurocholic acid | THCA | Ki | = | 39.4 | uM | ALA2077473 | 4.41 | inhibitor [Ki=39.4uM] | nM | Rattus norvegicus | |
| 5. |  ALA2074656 | N-retinyl-N-retinylidene ethanolamine | Ki | = | 37 | uM | ALA2078499 | 4.43 | inhibitor [Ki=37uM] | nM | Rattus norvegicus | |
| 6. |  ALA2074618 | Grapefruit juice | Activity | 0 | ALA2078497 | inhibitor [(at a rough estimate) 20 % of control] | Rattus norvegicus | |||||
| 7. |  ALA4297251 | Orange juice | Activity | 0 | ALA2078496 | inhibitor [(at a rough estimate) <5 % of control] | Rattus norvegicus | |||||
| 8. |  microcystin-LR | Microcystin-LR [4(E),6(Z)] | Activity | 0 | ALA2078419 | is not a substrate [(-)] | Rattus norvegicus | |||||
| 9. |  Quinine | 10a | Ki | = | 3.81 | uM | ALA2077474 | 5.42 | inhibitor [Ki=3.81uM] | nM | Rattus norvegicus | |
| 10. |  Ibuprofen | ibuprofen | Ki | = | 2430 | uM | ALA2077474 | inhibitor [Ki=2430uM] | nM | Rattus norvegicus | ||
| 11. | [³H]taurocholic acid | THCA | Ki | = | 156 | uM | ALA2078501 | inhibitor [Ki=156uM] | nM | Rattus norvegicus | ||
| 12. |  ALA2369946 | Demethylphalloin | Activity | 0 | ALA2078422 | is not a substrate [-] | Rattus norvegicus | |||||
| 13. |  ALA3527524 | N-methyl-quinidine | Activity | 0 | ALA2076302 | is not a substrate [-] | Rattus norvegicus | |||||
| 14. |  ALA2074787 | N-methyl-quinine | Activity | 0 | ALA2076302 | is not a substrate [-] | Rattus norvegicus | |||||
| 15. |  ALA2074720 | Bilirubin monoglucuronide | Activity | 0 | ALA2078131 | is not a substrate [-] | Rattus norvegicus | |||||
| 16. |  [³H]BSP | Bromosulfophthalein | Activity | 0 | ALA2078131 | is not a substrate [-] | Rattus norvegicus | |||||
| 17. |  ALA1201768 | Gadoxetate | Activity | 0 | ALA2078131 | is not a substrate [-] | Rattus norvegicus | |||||
| 18. |  ALA495936 | Leukotriene C4 (LTC4) | Activity | 0 | ALA2078131 | is not a substrate [-] | Rattus norvegicus | |||||
| 19. |  ALA2074644 | Taurolithocholate-3-sulfate | Activity | 0 | ALA2078131 | is not a substrate [-] | Rattus norvegicus | |||||
| 20. |  [³H]methotrexate | 138 | Activity | 0 | ALA2077065 | is not a substrate [-] | Rattus norvegicus |
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