# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PFI-3 | 72; PFI-3 | deltaTm | = | 7.5 | degrees C | ALA3790871 | degrees C | Homo sapiens | |||
2. | PFI-3 | 72; PFI-3 | Kd | = | 48 | nM | ALA3790868 | 7.32 | nM | Homo sapiens | ||
3. | ALA3774575 | 8i; IACS-9571 | Activity | > | 35 | % | ALA3777038 | % | Homo sapiens | |||
4. | ALA3774575 | 8i; IACS-9571 | Activity | > | 35 | % | ALA3777037 | % | Homo sapiens | |||
5. | GSK8573 | 23; GSK8573 | Activity | 0 | ALA3773276 | Not Active | Homo sapiens | |||||
6. | GSK 2801 | 1 | Activity | 0 | ALA3773276 | Not Active | Homo sapiens | |||||
7. | GSK8573 | 23; GSK8573 | Activity | 0 | ALA3773275 | Not Active | Homo sapiens | |||||
8. | GSK 2801 | 1 | Activity | 0 | ALA3773275 | Not Active | Homo sapiens | |||||
9. | GSK8573 | 23; GSK8573 | Activity | 0 | ALA3773274 | Not Active | Homo sapiens | |||||
10. | GSK 2801 | 1 | Activity | 0 | ALA3773274 | Not Active | Homo sapiens | |||||
11. | GSK8573 | 23; GSK8573 | Activity | 0 | ALA3773273 | Not Active | Homo sapiens | |||||
12. | GSK 2801 | 1 | Activity | 0 | ALA3773273 | Not Active | Homo sapiens | |||||
13. | GSK8573 | 23; GSK8573 | Activity | 0 | ALA3773272 | Not Active | Homo sapiens | |||||
14. | GSK 2801 | 1 | Activity | 0 | ALA3773272 | Not Active | Homo sapiens | |||||
15. | PFI-3 | 72; PFI-3 | Kd | = | 48 | nM | ALA3757231 | 7.32 | nM | Homo sapiens | ||
16. | PFI-3 | 72; PFI-3 | dTm | = | 9.1 | K | ALA5214137 | K | Homo sapiens | |||
17. | PFI-3 | 72; PFI-3 | Kd | = | 48 | nM | ALA5210532 | 7.32 | nM | Homo sapiens | ||
18. | PFI-3 | 72; PFI-3 | EC50 | < | 1000 | nM | ALA5210236 | nM | Homo sapiens | |||
19. | GNE-064 | 5; GNE-064 | Kd | = | 0.49 | uM | ALA5142218 | 6.31 | nM | Homo sapiens | ||
20. | PFI-3 | 72; PFI-3 | Kd | = | 5.8 | uM | ALA5142218 | 5.24 | nM | Homo sapiens |