# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | Kd | = | 190.1 | nM | ALA5210527 | 6.72 | nM | Homo sapiens | ||
2. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | IC50 | = | 4 | nM | ALA5210063 | 8.40 | nM | Homo sapiens | ||
3. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | IC50 | = | 4 | nM | ALA5210062 | 8.40 | nM | Homo sapiens | ||
4. | ALA5204783 | 8m | Kd | = | 194.9 | nM | ALA5162568 | 6.71 | nM | Homo sapiens | ||
5. | ALA5206088 | 8l; XY153 | Kd | = | 38.8 | nM | ALA5162568 | 7.41 | nM | Homo sapiens | ||
6. | ALA5204783 | 8m | Kd | = | 3308 | nM | ALA5162567 | 5.48 | nM | Homo sapiens | ||
7. | ALA5206088 | 8l; XY153 | Kd | = | 3668 | nM | ALA5162567 | 5.44 | nM | Homo sapiens | ||
8. | ALA5204783 | 8m | deltaTm | = | 11 | degrees C | ALA5162541 | degrees C | Homo sapiens | |||
9. | ALA5206088 | 8l; XY153 | deltaTm | = | 13.25 | degrees C | ALA5162541 | degrees C | Homo sapiens | |||
10. | ALA5205742 | 8k | deltaTm | = | 14.5 | degrees C | ALA5162541 | degrees C | Homo sapiens | |||
11. | ALA5178480 | 8j | deltaTm | = | 15 | degrees C | ALA5162541 | degrees C | Homo sapiens | |||
12. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | 11.25 | degrees C | ALA5162541 | degrees C | Homo sapiens | |||
13. | ALA5204783 | 8m | deltaTm | = | 2 | degrees C | ALA5162532 | degrees C | Homo sapiens | |||
14. | ALA5206088 | 8l; XY153 | deltaTm | = | 2 | degrees C | ALA5162532 | degrees C | Homo sapiens | |||
15. | ALA5205742 | 8k | deltaTm | = | 3 | degrees C | ALA5162532 | degrees C | Homo sapiens | |||
16. | ALA5178480 | 8j | deltaTm | = | 2.75 | degrees C | ALA5162532 | degrees C | Homo sapiens | |||
17. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | 5 | degrees C | ALA5162532 | degrees C | Homo sapiens | |||
18. | ALA5205457 | 3r; ZLD2218 | IC50 | > | 1 | uM | ALA5158666 | nM | Homo sapiens | |||
19. | ALA5195288 | 27 | pKd | = | 7.6 | ALA5157245 | 7.60 | nM | Homo sapiens | |||
20. | ALA5195288 | 27 | pKd | = | 7.6 | ALA5157244 | 7.60 | nM | Homo sapiens |