# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ARV-771 | 5 | DC50 | < | 1 | nM | ALA5246315 | nM | Homo sapiens | |||
2. | ALA5283149 | 43 | DC50 | = | 25 | nM | ALA5243399 | nM | Homo sapiens | |||
3. | ARV-771 | 5 | DC50 | < | 5 | nM | ALA5243383 | nM | Homo sapiens | |||
4. | ARV-771 | 5 | DC50 | < | 5 | nM | ALA5243382 | nM | Homo sapiens | |||
5. | ARV-771 | 5 | DC50 | < | 5 | nM | ALA5243381 | nM | Homo sapiens | |||
6. | Mz1 | 1; MZ-1 | Kd | = | 115 | nM | ALA5243376 | 6.94 | nM | Homo sapiens | ||
7. | ALA2393130 | RVX-208 | IC50 | = | 0.51 | uM | ALA5242785 | 6.29 | nM | Homo sapiens | ||
8. | ALA2393130 | RVX-208 | IC50 | = | 87 | uM | ALA5242784 | 4.06 | nM | Homo sapiens | ||
9. | ALA5274024 | 41; NEO2734 | Kd | = | 3.5 | nM | ALA5241956 | 8.46 | nM | Homo sapiens | ||
10. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | 10 | degrees C | ALA5236402 | degrees C | Homo sapiens | |||
11. | ALA5267793 | 9d | deltaTm | = | 2.3 | degrees C | ALA5236402 | degrees C | Homo sapiens | |||
12. | ALA2017287 | 34 | Kd | = | 32 | nM | ALA5232443 | 7.50 | nM | Homo sapiens | ||
13. | OTX015 | 4, OTX015 | IC50 | = | 92 | nM | ALA5231287 | 7.04 | nM | Homo sapiens | ||
14. | ARV-771 | 5 | Kd | = | 7.6 | nM | ALA5231278 | 8.12 | nM | Homo sapiens | ||
15. | ALA5281933 | 12d; AT1 | Kd | = | 39 | nM | ALA5231278 | 7.41 | nM | Homo sapiens | ||
16. | Mz1 | 1; MZ-1 | Kd | = | 115 | nM | ALA5231278 | 6.94 | nM | Homo sapiens | ||
17. | ARV-771 | 5 | Kd | = | 8.3 | nM | ALA5231277 | 8.08 | nM | Homo sapiens | ||
18. | ALA5281933 | 12d; AT1 | Kd | = | 35 | nM | ALA5231277 | 7.46 | nM | Homo sapiens | ||
19. | Mz1 | 1; MZ-1 | Kd | = | 119 | nM | ALA5231277 | 6.92 | nM | Homo sapiens | ||
20. | ALA5279987 | 26; SIM1 | DC50 | = | 3.3 | nM | ALA5224301 | nM | Homo sapiens |