# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AAPK-25 | AAPK-25 | Kd | = | 8.02 | uM | ALA4375313 | 5.10 | nM | Homo sapiens | ||
2. | ALA4084955 | 14 | INH | = | -8.2 | % | ALA4034286 | % | Homo sapiens | |||
3. | OSI-930 | OSI-930 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
4. | PF-562271 | PF-562271 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
5. | Sotrastaurin | 1 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
6. | SNS-032 (BMS-387032) | 21 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
7. | LY2603618 | RABUSERTIB | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
8. | CEP-32496 | 40, CEP-32496 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
9. | Roscovitine (Seliciclib,CYC202) | Roscovitine | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
10. | ALA1233528 | VOLASERTIB | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
11. | BI 2536 | 1 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
12. | Regorafenib (BAY 73-4506) | 2, BAY-734506 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
13. | ALA3545137 | PF-00477736 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
14. | LY2801653 | MERESTINIB | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
15. | ALA502835 | 3, BIBF1120 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
16. | Sunitinib | 12b | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
17. | Amuvatinib (MP-470) | AMUVATINIB | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
18. | Pelitinib | EKB-569 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
19. | Entrectinib | SID103905026 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens | ||
20. | PF-3758309 | 1, PF-3758309 | Kd apparent | > | 30000 | nM | ALA3991651 | Inactive | nM | Homo sapiens |