# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4802048 | EUB0001565 | IC50 | 271 | nM | ALA4887759 | Not Active | nM | Homo sapiens | |||
2. | BAY-091 | EUB0001564 | EC50 | 1.1 | uM | ALA4887761 | Active | nM | Homo sapiens | |||
3. | BAY-091 | EUB0001564 | EC50 | 1.8 | uM | ALA4887760 | Active | nM | Homo sapiens | |||
4. | BAY-091 | EUB0001564 | IC50 | 21 | nM | ALA4887759 | Active | nM | Homo sapiens | |||
5. | BAY-091 | EUB0001564 | IC50 | 16.4 | nM | ALA4887758 | Active | nM | Homo sapiens | |||
6. | BAY-091 | EUB0001564 | IC50 | 8.5 | nM | ALA4887757 | Active | nM | Homo sapiens | |||
7. | BAY-091 | EUB0001564 | IC50 | 2.6 | nM | ALA4887756 | Active | nM | Homo sapiens | |||
8. | BAY-091 | EUB0001564 | IC50 | 1.3 | nM | ALA4887755 | Active | nM | Homo sapiens | |||
9. | BAY-091 | EUB0001564 | % inhibition | 142.02 | % | ALA4888004 | Not Active | % | Homo sapiens | |||
10. | BI 605906 | BI605906 | % Ctrl | 115 | % | ALA4887307 | Not Active | % | Homo sapiens | |||
11. | ALA4580220 | EUB0000311 | % residual kinase activity | 105 | % | ALA4884537 | Not Active | % | Homo sapiens | |||
12. | BAY-885 | BAY-885; 41 | % residual kinase activity | 95 | % | ALA4881299 | Not Active | % | Homo sapiens | |||
13. | ALA4561692 | 1 | pIC50 | < | 5 | ALA4479386 | nM | Homo sapiens | ||||
14. | ALA4859660 | I-9 | INH | = | 0 | % | ALA4804651 | % | Homo sapiens | |||
15. | ALA4868141 | I-65 | INH | = | 0 | % | ALA4804651 | % | Homo sapiens | |||
16. | ALA4855730 | I-51 | INH | = | 0 | % | ALA4804651 | % | Homo sapiens | |||
17. | ALA4867931 | I-50 | INH | > | 90 | % | ALA4804651 | % | Homo sapiens | |||
18. | ALA4860979 | I-28 | INH | = | 0 | % | ALA4804651 | % | Homo sapiens | |||
19. | ALA4855542 | I-13 | INH | = | 0 | % | ALA4804651 | % | Homo sapiens | |||
20. | ALA4859660 | I-9 | % inhibition | = | 10.2 | uM | ALA4804469 | Data is reported as I50 but values are consistent with % inhibition, changed for ChEMBL32 at suggestion of BZ | uM | Homo sapiens |