| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  (5Z)-7-Oxozeaenol | 1, f152A1 | INH | = | -47.8 | % | ALA4118476 | % | Homo sapiens | |||
| 2. |  N-{2-[(5-chloro-2-{[1-(2-methoxyethyl)-1H-pyrazol-4-yl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | 25 | INH | = | -31.3 | % | ALA4118476 | % | Homo sapiens | |||
| 3. |  SM1-71 | 5 | INH | = | -77 | % | ALA4118476 | % | Homo sapiens | |||
| 4. |  ALA3971067 | BDBM223552 | INH | = | 26.2 | % | ALA4046084 | % | Homo sapiens | |||
| 5. | ALA3971067 | BDBM223552 | INH | = | -9.8 | % | ALA4046083 | % | Homo sapiens | |||
| 6. | ALA3971067 | BDBM223552 | INH | = | 8.7 | % | ALA4045843 | % | Homo sapiens | |||
| 7. | ALA3971067 | BDBM223552 | INH | = | -61.1 | % | ALA4045842 | % | Homo sapiens | |||
| 8. |  ALA4084955 | 14 | INH | = | 5.4 | % | ALA4034497 | % | Homo sapiens | |||
| 9. |  GSK1059615 | GSK-1059615 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 10. |  RAF265 (CHIR-265) | CHIR-265/RAF-265 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 11. |  TAK-285 | 34e, TAK-285 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 12. |  6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine | 14, ENMD-2076 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 13. |  LY2801653 | MERESTINIB | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 14. |  Canertinib (CI-1033) | 18 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 15. |  AT9283 | 16, AT9283 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 16. |  TG02 (Double bond E) | 26h, SB1317/TG02 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 17. |  AZD1152 | 5 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 18. |  Lenvatinib (E7080) | E7080 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 19. |  CP-724714 | 4 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens | ||
| 20. |  ALA608533 | PKC-412 | Kd apparent | > | 30000 | nM | ALA3991899 | Inactive | nM | Homo sapiens |
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