# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5219936 | RgIA-5474 | IC50 | > | 10000 | nM | ALA5215844 | nM | Rattus norvegicus | |||
2. | ALA4540592 | 14; [C2S,C9S,C20A,C27A]GeXIVA | IC50 | = | 3710 | nM | ALA4381859 | 5.43 | nM | Rattus norvegicus | ||
3. | ALA4460411 | 13; [C2A,C9A,C20S,C27S]GeXIVA | IC50 | = | 2830 | nM | ALA4381859 | 5.55 | nM | Rattus norvegicus | ||
4. | ALA4448288 | 12; [C2S,C9S,C20S,C27S]GeXIVA | IC50 | = | 2090 | nM | ALA4381859 | 5.68 | nM | Rattus norvegicus | ||
5. | ALA4463717 | 11; [C2A,C9A,C20A,C27A]GeXIVA | IC50 | = | 3570 | nM | ALA4381859 | 5.45 | nM | Rattus norvegicus | ||
6. | ALA4554920 | 10; [C9S,C20S]GeXIVA[1,4] | IC50 | = | 1180 | nM | ALA4381859 | 5.93 | nM | Rattus norvegicus | ||
7. | ALA4473421 | 9; [C9A,C20A]GeXIVA[1,4] | IC50 | = | 1050 | nM | ALA4381859 | 5.98 | nM | Rattus norvegicus | ||
8. | ALA4455583 | 8; [C2S,C27S]GeXIVA[1,4] | IC50 | = | 1570 | nM | ALA4381859 | 5.80 | nM | Rattus norvegicus | ||
9. | ALA4577696 | 7; [C2A,C27A]GeXIVA[1,4] | IC50 | = | 1370 | nM | ALA4381859 | 5.86 | nM | Rattus norvegicus | ||
10. | ALA4553407 | 6; GeXIVA[1,4] | IC50 | = | 1250 | nM | ALA4381859 | 5.90 | nM | Rattus norvegicus | ||
11. | ALA4450578 | 5; [C20S,C27S]GeXIVA[1,2] | IC50 | = | 2780 | nM | ALA4381859 | 5.56 | nM | Rattus norvegicus | ||
12. | ALA4522506 | 4; [C20A,C27A]GeXIVA[1,2] | IC50 | = | 3250 | nM | ALA4381859 | 5.49 | nM | Rattus norvegicus | ||
13. | ALA4525995 | 3; [C2S,C9S]GeXIVA[1,2] | IC50 | = | 3800 | nM | ALA4381859 | 5.42 | nM | Rattus norvegicus | ||
14. | ALA4446775 | 2; [C2A,C9A]GeXIVA[1,2] | IC50 | = | 4740 | nM | ALA4381859 | 5.32 | nM | Rattus norvegicus | ||
15. | ALA4460879 | 1; GeXIVA[1,2] | IC50 | = | 940 | nM | ALA4381859 | 6.03 | nM | Rattus norvegicus | ||
16. | ALA4869892 | PeIA-5667 | INH | = | 94 | % | ALA4811761 | % | Rattus norvegicus | |||
17. | ALA4865866 | PeIA-5069 | IC50 | > | 10000 | nM | ALA4811720 | nM | Rattus norvegicus | |||
18. | ALA4871260 | [Ala4,Hyp5]BuIA | IC50 | > | 10000 | nM | ALA4811720 | nM | Rattus norvegicus | |||
19. | ALA4867647 | [Ala9,Ala15]MII | IC50 | = | 4850 | nM | ALA4811720 | 5.31 | nM | Rattus norvegicus | ||
20. | ALA4872191 | PeIA-5712 | IC50 | = | 9505 | nM | ALA4811720 | 5.02 | nM | Rattus norvegicus |