# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5219936 | RgIA-5474 | IC50 | > | 10000 | nM | ALA5215850 | nM | Rattus norvegicus | |||
2. | ALA4540592 | 14; [C2S,C9S,C20A,C27A]GeXIVA | IC50 | = | 4900 | nM | ALA4381861 | 5.31 | nM | Rattus norvegicus | ||
3. | ALA4460411 | 13; [C2A,C9A,C20S,C27S]GeXIVA | IC50 | = | 4360 | nM | ALA4381861 | 5.36 | nM | Rattus norvegicus | ||
4. | ALA4448288 | 12; [C2S,C9S,C20S,C27S]GeXIVA | IC50 | = | 7520 | nM | ALA4381861 | 5.12 | nM | Rattus norvegicus | ||
5. | ALA4463717 | 11; [C2A,C9A,C20A,C27A]GeXIVA | IC50 | = | 7510 | nM | ALA4381861 | 5.12 | nM | Rattus norvegicus | ||
6. | ALA4554920 | 10; [C9S,C20S]GeXIVA[1,4] | IC50 | = | 2160 | nM | ALA4381861 | 5.67 | nM | Rattus norvegicus | ||
7. | ALA4473421 | 9; [C9A,C20A]GeXIVA[1,4] | IC50 | = | 3980 | nM | ALA4381861 | 5.40 | nM | Rattus norvegicus | ||
8. | ALA4455583 | 8; [C2S,C27S]GeXIVA[1,4] | IC50 | = | 2230 | nM | ALA4381861 | 5.65 | nM | Rattus norvegicus | ||
9. | ALA4577696 | 7; [C2A,C27A]GeXIVA[1,4] | IC50 | = | 2990 | nM | ALA4381861 | 5.52 | nM | Rattus norvegicus | ||
10. | ALA4553407 | 6; GeXIVA[1,4] | IC50 | = | 440 | nM | ALA4381861 | 6.36 | nM | Rattus norvegicus | ||
11. | ALA4450578 | 5; [C20S,C27S]GeXIVA[1,2] | IC50 | = | 9120 | nM | ALA4381861 | 5.04 | nM | Rattus norvegicus | ||
12. | ALA4522506 | 4; [C20A,C27A]GeXIVA[1,2] | IC50 | = | 3120 | nM | ALA4381861 | 5.51 | nM | Rattus norvegicus | ||
13. | ALA4525995 | 3; [C2S,C9S]GeXIVA[1,2] | IC50 | = | 9060 | nM | ALA4381861 | 5.04 | nM | Rattus norvegicus | ||
14. | ALA4446775 | 2; [C2A,C9A]GeXIVA[1,2] | IC50 | = | 9450 | nM | ALA4381861 | 5.03 | nM | Rattus norvegicus | ||
15. | ALA4460879 | 1; GeXIVA[1,2] | IC50 | = | 1610 | nM | ALA4381861 | 5.79 | nM | Rattus norvegicus | ||
16. | ALA4872191 | PeIA-5712 | INH | = | 77 | % | ALA4811759 | % | Rattus norvegicus | |||
17. | ALA4869892 | PeIA-5667 | INH | = | 98 | % | ALA4811759 | % | Rattus norvegicus | |||
18. | ALA4872191 | PeIA-5712 | IC50 | > | 10000 | nM | ALA4811716 | nM | Rattus norvegicus | |||
19. | ALA4869892 | PeIA-5667 | IC50 | > | 10000 | nM | ALA4811716 | nM | Rattus norvegicus | |||
20. | ALA4215824 | 12 | INH | < | 50 | % | ALA4202189 | % | Rattus norvegicus |