# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5219936 | RgIA-5474 | IC50 | > | 10000 | nM | ALA5215855 | nM | Rattus norvegicus | |||
2. | ALA5186760 | 16 | Ki | = | 81.55 | uM | ALA5147132 | 4.09 | nM | Rattus norvegicus | ||
3. | ALA5200745 | 15 | Ki | > | 100 | uM | ALA5147132 | nM | Rattus norvegicus | |||
4. | ALA5178221 | 14 | Ki | > | 100 | uM | ALA5147132 | nM | Rattus norvegicus | |||
5. | ALA5200048 | 13 | Ki | = | 27.1 | uM | ALA5147132 | 4.57 | nM | Rattus norvegicus | ||
6. | ALA5183330 | 12 | Ki | = | 45.31 | uM | ALA5147132 | 4.34 | nM | Rattus norvegicus | ||
7. | ALA433777 | 13 | Ki | = | 19.43 | uM | ALA5147132 | 4.71 | nM | Rattus norvegicus | ||
8. | ALA4531337 | 8ai | Emax | = | 78 | % | ALA4390087 | % | Rattus norvegicus | |||
9. | ALA4540592 | 14; [C2S,C9S,C20A,C27A]GeXIVA | IC50 | = | 5750 | nM | ALA4381860 | 5.24 | nM | Rattus norvegicus | ||
10. | ALA4460411 | 13; [C2A,C9A,C20S,C27S]GeXIVA | IC50 | = | 8350 | nM | ALA4381860 | 5.08 | nM | Rattus norvegicus | ||
11. | ALA4448288 | 12; [C2S,C9S,C20S,C27S]GeXIVA | IC50 | = | 6630 | nM | ALA4381860 | 5.18 | nM | Rattus norvegicus | ||
12. | ALA4463717 | 11; [C2A,C9A,C20A,C27A]GeXIVA | IC50 | = | 8990 | nM | ALA4381860 | 5.05 | nM | Rattus norvegicus | ||
13. | ALA4554920 | 10; [C9S,C20S]GeXIVA[1,4] | IC50 | = | 3660 | nM | ALA4381860 | 5.44 | nM | Rattus norvegicus | ||
14. | ALA4473421 | 9; [C9A,C20A]GeXIVA[1,4] | IC50 | = | 4750 | nM | ALA4381860 | 5.32 | nM | Rattus norvegicus | ||
15. | ALA4455583 | 8; [C2S,C27S]GeXIVA[1,4] | IC50 | = | 7570 | nM | ALA4381860 | 5.12 | nM | Rattus norvegicus | ||
16. | ALA4577696 | 7; [C2A,C27A]GeXIVA[1,4] | IC50 | = | 6310 | nM | ALA4381860 | 5.20 | nM | Rattus norvegicus | ||
17. | ALA4553407 | 6; GeXIVA[1,4] | IC50 | = | 3400 | nM | ALA4381860 | 5.47 | nM | Rattus norvegicus | ||
18. | ALA4450578 | 5; [C20S,C27S]GeXIVA[1,2] | IC50 | = | 4280 | nM | ALA4381860 | 5.37 | nM | Rattus norvegicus | ||
19. | ALA4522506 | 4; [C20A,C27A]GeXIVA[1,2] | IC50 | = | 6130 | nM | ALA4381860 | 5.21 | nM | Rattus norvegicus | ||
20. | ALA4525995 | 3; [C2S,C9S]GeXIVA[1,2] | IC50 | = | 8410 | nM | ALA4381860 | 5.08 | nM | Rattus norvegicus |