# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | MRK 016 | 13 | EC50 | = | 15 | ng/ml | ALA5242037 | ug.mL-1 | Rattus norvegicus | |||
2. | ALA5273865 | 41 | IC50 | = | 2 | nM | ALA5237498 | 8.70 | nM | Rattus norvegicus | ||
3. | ALA5284940 | 40 | INH | = | 80 | % | ALA5237497 | % | Rattus norvegicus | |||
4. | ALA5274306 | 15 | INH | < | 50 | % | ALA5228830 | % | Rattus norvegicus | |||
5. | ALA5174845 | rac-1f | INH | < | 50 | % | ALA5123263 | % | Rattus norvegicus | |||
6. | ALA5175769 | rac-1d | INH | < | 50 | % | ALA5123263 | % | Rattus norvegicus | |||
7. | ALA5198193 | 1c | IC50 | = | 23 | nM | ALA5123262 | 7.64 | nM | Rattus norvegicus | ||
8. | ALA1468243 | SID14727391 | IC50 | = | 1.94 | nM | ALA5123262 | 8.71 | nM | Rattus norvegicus | ||
9. | ALA5175769 | rac-1d | IC50 | = | 34 | nM | ALA5123262 | 7.47 | nM | Rattus norvegicus | ||
10. | ALA5175769 | rac-1d | IC50 | = | 10.9 | nM | ALA5123262 | 7.96 | nM | Rattus norvegicus | ||
11. | ALA5174845 | rac-1f | IC50 | = | 430 | nM | ALA5123262 | 6.37 | nM | Rattus norvegicus | ||
12. | ALA5174845 | rac-1f | IC50 | = | 210 | nM | ALA5123262 | 6.68 | nM | Rattus norvegicus | ||
13. | Diazepam | Diazepam | IC50 | = | 16 | nM | ALA5123262 | 7.80 | nM | Rattus norvegicus | ||
14. | Clarithromycin | clarithromycin | Ki | > | 10 | uM | ALA4432806 | nM | Rattus norvegicus | |||
15. | Clarithromycin | clarithromycin | INH | 0 | ALA4432813 | Not Active | % | Rattus norvegicus | ||||
16. | Clarithromycin | clarithromycin | Kd | = | 0.64 | nM | ALA4432812 | 9.19 | nM | Rattus norvegicus | ||
17. | ALA2334661 | 14a | INH | = | 6 | % | ALA4421239 | % | Rattus norvegicus | |||
18. | ALA2334661 | 14a | INH | = | -6 | % | ALA4421238 | % | Rattus norvegicus | |||
19. | ALA2203406 | 17, CJ-1639 | INH | < | 50 | % | ALA4406673 | % | Rattus norvegicus | |||
20. | Pramipexole | (-)-2 | INH | 0 | ALA4406673 | Not Determined | % | Rattus norvegicus |