# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3113642 | 16 | INH | = | 4 | % | ALA3117961 | % | Rattus norvegicus | |||
2. | ALA3113644 | 18 | INH | = | 4 | % | ALA3117960 | % | Rattus norvegicus | |||
3. | BI 605906 | BI605906 | % Ctrl | 93 | % | ALA4887175 | Not Active | % | Rattus norvegicus | |||
4. | BI 605906 | BI605906 | % Ctrl | 109 | % | ALA4887175 | Not Active | % | Rattus norvegicus | |||
5. | BI-1950 | EUB0000310 | % Ctrl | 102 | % | ALA4887060 | Not Active | % | Rattus norvegicus | |||
6. | 5-[2-[5-chloro-2-[(5-ethoxyquinolin-8-yl)sulfonylamino]phenyl]ethynyl]-4-methoxypyridine-2-carboxylic acid | EUB0001566 | % Inhibition of Control Specific Binding (Mean n=2) | 6.6 | % | ALA4886134 | % | Rattus norvegicus | ||||
7. | BI-1935 | EUB0000542 | % Ctrl | 94 | % | ALA4882489 | Not Active | % | Rattus norvegicus | |||
8. | BI 653048 | (R)-39 | % Ctrl | 89 | % | ALA4882192 | Not Active | % | Rattus norvegicus | |||
9. | ALA3688396 | BDBM168626 | IC50 | = | 100 | nM | ALA3706372 | 7.00 | 312560 | nM | Rattus norvegicus | |
10. | ALA3688395 | BDBM168625 | IC50 | = | 150 | nM | ALA3706372 | 6.82 | 312559 | nM | Rattus norvegicus | |
11. | ALA3688394 | BDBM168624 | IC50 | = | 100 | nM | ALA3706372 | 7.00 | 312558 | nM | Rattus norvegicus | |
12. | ALA3688393 | BDBM168622 | IC50 | = | 350 | nM | ALA3706372 | 6.46 | 312557 | nM | Rattus norvegicus | |
13. | ALA3688392 | BDBM168621 | IC50 | = | 350 | nM | ALA3706372 | 6.46 | 312556 | nM | Rattus norvegicus | |
14. | ALA3688391 | BDBM168620 | IC50 | = | 300 | nM | ALA3706372 | 6.52 | 312555 | nM | Rattus norvegicus | |
15. | ALA3688390 | BDBM168619 | IC50 | = | 340 | nM | ALA3706372 | 6.47 | 312554 | nM | Rattus norvegicus | |
16. | ALA3688389 | BDBM168618 | IC50 | = | 350 | nM | ALA3706372 | 6.46 | 312553 | nM | Rattus norvegicus | |
17. | ALA3688388 | BDBM168617 | IC50 | = | 620 | nM | ALA3706372 | 6.21 | 312552 | nM | Rattus norvegicus | |
18. | ALA3683711 | BDBM168616 | IC50 | = | 720 | nM | ALA3706372 | 6.14 | 312551 | nM | Rattus norvegicus | |
19. | Phentolamine | Phentolamine | Ki | = | 10.3 | nM | ALA3240449 | 7.99 | nM | Rattus norvegicus | ||
20. | ALA3233679 | 25a | Ki | = | 181.1 | nM | ALA3240449 | 6.74 | nM | Rattus norvegicus |