# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3775181 | 3d | IC50 | < | 5 | uM | ALA3778052 | nM | Homo sapiens | |||
2. | ALA3745885 | 7ao; ON1231320 | IC50 | > | 10 | uM | ALA3750029 | nM | Homo sapiens | |||
3. | ALA3628628 | 5 | INH | = | -4.89 | % | ALA3631114 | % | Homo sapiens | |||
4. | ALA3628627 | 4 | INH | = | 24.99 | % | ALA3631114 | % | Homo sapiens | |||
5. | ALA166031 | 3 | INH | = | -0.31 | % | ALA3631114 | % | Homo sapiens | |||
6. | ALA5177284 | 10w | Kd | = | 670 | nM | ALA5136618 | 6.17 | nM | Homo sapiens | ||
7. | ALA4206831 | 2; FMF-03-145-1 | Activity | = | 68 | % | ALA4186033 | % | Homo sapiens | |||
8. | ALA3969370 | 19; FMF-01-086-2 | Activity | = | 96 | % | ALA4186033 | % | Homo sapiens | |||
9. | ALA4174988 | 15i | Activity | = | 92 | % | ALA4157254 | % | Homo sapiens | |||
10. | ALA4080797 | 35 | Activity | = | 74 | % | ALA4055099 | % | Homo sapiens | |||
11. | ALA4096145 | 2 | Activity | = | 92 | % | ALA4055099 | % | Homo sapiens | |||
12. | ALA4092508 | 2t | Activity | = | 100 | % | ALA4044175 | % | Homo sapiens | |||
13. | ALA4533018 | IM-93 | Activity | = | 100 | % | ALA4308031 | % | Homo sapiens | |||
14. | JSH-150 | 40; JSH-150 | Activity | = | 95 | % | ALA4264522 | % | Homo sapiens | |||
15. | PDGFRα kinase inhibitor 1 | 15i | Activity | = | 81 | % | ALA4230933 | % | Homo sapiens | |||
16. | ALA4077123 | 9; CHMFL-BTK-01 | Activity | = | 90 | % | ALA4025364 | % | Homo sapiens | |||
17. | GSK 114 | 2 | INH | = | 3 | % | ALA3816763 | % | Homo sapiens | |||
18. | Staurosporine | 1 (Staurosporine) | IC50 | = | 6.9 | 10'-8M | ALA4412098 | 7.16 | nM | Homo sapiens | ||
19. | ALA4476753 | 1n | Activity | = | 58.59 | % | ALA4412082 | % | Homo sapiens | |||
20. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405546 | % | Homo sapiens |