# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3409970 | 20 | INH | 0 | ALA3414097 | Active | % | Homo sapiens | ||||
2. | ALA3409969 | 19 | Ratio | = | 82000 | /M/min | ALA3413585 | /M/min | Homo sapiens | |||
3. | ALA4464539 | 2 | IC50 | = | 80 | uM | ALA4433158 | 4.10 | nM | Homo sapiens | ||
4. | ALA4442207 | 6 | IC50 | > | 500 | uM | ALA4433158 | nM | Homo sapiens | |||
5. | ALA4461562 | 7 | IC50 | = | 52 | uM | ALA4433158 | 4.28 | nM | Homo sapiens | ||
6. | ALA4473416 | 10 | IC50 | = | 125 | uM | ALA4433158 | nM | Homo sapiens | |||
7. | ALA4546087 | 13 | IC50 | = | 408 | uM | ALA4433158 | nM | Homo sapiens | |||
8. | ALA4468883 | 18 | IC50 | = | 34 | uM | ALA4433158 | 4.47 | nM | Homo sapiens | ||
9. | ALA4449566 | 20 | IC50 | = | 161 | uM | ALA4433158 | nM | Homo sapiens | |||
10. | ALA4547728 | 23 | IC50 | = | 294 | uM | ALA4433158 | nM | Homo sapiens | |||
11. | ALA1962723 | L-F-amidine | Ratio | = | 2800 | /M/min | ALA2212942 | /M/min | Homo sapiens | |||
12. | ALA1962361 | L-Cl-amidine | Ratio | = | 37000 | /M/min | ALA2212942 | /M/min | Homo sapiens | |||
13. | ALA1962643 | L-o-F-amidine | Ratio | = | 180851 | /M/min | ALA2212942 | /M/min | Homo sapiens | |||
14. | ALA2204312 | D-F-amidine | Ratio | = | 1220 | /M/min | ALA2212942 | /M/min | Homo sapiens | |||
15. | ALA2204313 | D-Cl-amidine | Ratio | = | 13500 | /M/min | ALA2212942 | /M/min | Homo sapiens | |||
16. | ALA2204314 | D-o-F-amidine | Ratio | = | 12100 | /M/min | ALA2212942 | /M/min | Homo sapiens | |||
17. | ALA2204315 | D-o-Cl-amidine | Ratio | = | 125 | /M/min | ALA2212942 | /M/min | Homo sapiens | |||
18. | ALA2204967 | D-Cl-amidine-Gly | Ratio | = | 190 | /M/min | ALA2212942 | /M/min | Homo sapiens | |||
19. | ALA2204968 | D-Cl-amidine-OH | Ratio | = | 230 | /M/min | ALA2212942 | /M/min | Homo sapiens | |||
20. | ALA2204969 | D-Cl2-amidine | Ratio | = | 150 | /M/min | ALA2212942 | /M/min | Homo sapiens |