# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3403619 | 22b, enantiomer-2 | Emax | = | 104 | % | ALA3404802 | % | Mus musculus | |||
2. | ALA3403619 | 22b, enantiomer-2 | EC50 | = | 0.05 | nM | ALA3404801 | 10.30 | nM | Mus musculus | ||
3. | ALA3359523 | 25 | Emax | = | 95 | % | ALA3380158 | % | Mus musculus | |||
4. | ALA3359522 | 24 | Emax | = | 104 | % | ALA3380158 | % | Mus musculus | |||
5. | ALA3359523 | 25 | EC50 | = | 0.064 | nM | ALA3380157 | 10.19 | nM | Mus musculus | ||
6. | ALA3359522 | 24 | EC50 | = | 0.05 | nM | ALA3380157 | 10.30 | nM | Mus musculus | ||
7. | etrasimod | (R)-4, APD334 | EC50 | = | 0.44 | nM | ALA3380990 | 9.36 | nM | Mus musculus | ||
8. | etrasimod | (R)-4, APD334 | Emax | = | 95 | % | ALA3380991 | % | Mus musculus | |||
9. | ALA3605533 | 21 | INH | 0 | ALA3607262 | Active | % | Mus musculus | ||||
10. | ALA3605516 | 4 | INH | 0 | ALA3607262 | Active | % | Mus musculus | ||||
11. | ALA3908980 | BDBM221929 | EC50 | = | 14.3 | nM | ALA3888306 | 7.84 | 388416 | nM | Mus musculus | |
12. | ALA3933363 | BDBM221928 | EC50 | = | 9.9 | nM | ALA3888306 | 8.00 | 388415 | nM | Mus musculus | |
13. | ALA3945798 | BDBM221926 | EC50 | = | 20 | nM | ALA3888306 | 7.70 | 388414 | nM | Mus musculus | |
14. | ALA3932290 | BDBM221923 | EC50 | = | 354 | nM | ALA3888306 | 6.45 | 388413 | nM | Mus musculus | |
15. | ALA3916072 | BDBM221932 | EC50 | = | 8 | nM | ALA3888306 | 8.10 | 388412 | nM | Mus musculus | |
16. | ALA3892404 | BDBM221916 | EC50 | = | 27 | nM | ALA3888306 | 7.57 | 388411 | nM | Mus musculus | |
17. | ALA3897804 | BDBM221914 | EC50 | = | 3.1 | nM | ALA3888306 | 8.51 | 388410 | nM | Mus musculus | |
18. | ALA3934780 | BDBM221913 | EC50 | = | 77 | nM | ALA3888306 | 7.11 | 388409 | nM | Mus musculus | |
19. | ALA2048293 | 23 | EC50 | = | 0.52 | nM | ALA2049907 | 9.28 | nM | Mus musculus | ||
20. | ALA2048293 | 23 | EC50 | = | 5.5 | nM | ALA2049907 | 8.26 | nM | Mus musculus |