# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ML348 | GNF-Pf-1127 | IC50 | > | 10 | uM | ALA3215055 | inactive | nM | Homo sapiens | ||
2. | ALA1673415 | Palmostatin B | IC50 | = | 37.7 | nM | ALA3135194 | 7.42 | nM | Homo sapiens | ||
3. | ALA3133031 | Palmostatin M | IC50 | = | 19.6 | nM | ALA3135194 | 7.71 | nM | Homo sapiens | ||
4. | ALA3133032 | Compound 4 | Ki | = | 0.73 | uM | ALA3135192 | 6.14 | nM | Homo sapiens | ||
5. | ALA1903566 | SID99445338 | IC50 | = | 30 | nM | ALA3135191 | 7.52 | nM | Homo sapiens | ||
6. | ALA3133033 | AA401 | IC50 | = | 200 | nM | ALA3135191 | 6.70 | nM | Homo sapiens | ||
7. | ALA1891894 | SID99445332 | IC50 | > | 1 | 10'4nM | ALA3135191 | nM | Homo sapiens | |||
8. | ML348 | GNF-Pf-1127 | Ki | > | 10 | uM | ALA3135187 | nM | Homo sapiens | |||
9. | ML 349 | SID24812860 | Ki | = | 230 | nM | ALA3135187 | 6.64 | nM | Homo sapiens | ||
10. | ALA1673415 | Palmostatin B | Ki | = | 34 | nM | ALA3135194 | 7.47 | nM | Homo sapiens | ||
11. | ALA3944678 | ML349-biotin | Activity | 0 | ALA3879679 | Active | Homo sapiens | |||||
12. | ML 349 | SID24812860 | Activity | 0 | ALA3879679 | Active | Homo sapiens | |||||
13. | ALA3944678 | ML349-biotin | IC50 | > | 10 | uM | ALA3879677 | nM | Homo sapiens | |||
14. | ML 349 | SID24812860 | IC50 | = | 1.1 | uM | ALA3879677 | 5.96 | nM | Homo sapiens | ||
15. | ALA3944678 | ML349-biotin | Activity | 0 | ALA3879676 | Homo sapiens | ||||||
16. | ALA3944678 | ML349-biotin | FC | > | 5 | ALA3879669 | Homo sapiens | |||||
17. | ALA3944678 | ML349-biotin | FC | > | 5 | ALA3879663 | Homo sapiens | |||||
18. | Azide-PEG3-biotin conjugate | Azide-PEG3-biotin | Activity | 0 | ALA3879662 | Homo sapiens | ||||||
19. | ALA3917640 | o-ML349-biotin | Activity | 0 | ALA3879662 | Homo sapiens | ||||||
20. | ALA3944678 | ML349-biotin | Activity | 0 | ALA3879662 | Active | Homo sapiens |