# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3086655 | 17 | t1/2 | = | 0.4 | hr | ALA3091130 | hr | Sus scrofa | |||
2. | ALA3086654 | 18 | Stability | 0 | ALA3091128 | Stable | % | Sus scrofa | ||||
3. | ALA3086653 | 19 | Stability | 0 | ALA3091128 | Stable | % | Sus scrofa | ||||
4. | ALA410972 | 1 | Stability | 0 | ALA3091127 | Unstable | % | Sus scrofa | ||||
5. | ALA3086850 | 8 | Stability | 0 | ALA3091124 | Stable | % | Sus scrofa | ||||
6. | ALA2315239 | 4.3TFA | Ki | = | 62.6 | nM | ALA2320210 | 7.20 | nM | Sus scrofa | ||
7. | ALA2315240 | 5.TFA | Ki | = | 3.4 | nM | ALA2320210 | 8.47 | nM | Sus scrofa | ||
8. | ALA2315241 | 6.TFA | Ki | = | 19.4 | nM | ALA2320210 | 7.71 | nM | Sus scrofa | ||
9. | ALA2315242 | 7.TFA | Ki | = | 7.8 | nM | ALA2320210 | 8.11 | nM | Sus scrofa | ||
10. | ALA2315243 | 8.3TFA | Ki | = | 38.3 | nM | ALA2320210 | 7.42 | nM | Sus scrofa | ||
11. | ALA2315244 | 9.TFA | Ki | = | 24.9 | nM | ALA2320210 | 7.60 | nM | Sus scrofa | ||
12. | ALA2315245 | 10.TFA | Ki | = | 0.6 | nM | ALA2320210 | 9.22 | nM | Sus scrofa | ||
13. | ALA2315246 | 11.TFA | Ki | = | 3 | nM | ALA2320210 | 8.52 | nM | Sus scrofa | ||
14. | ALA2315247 | 12.TFA | Ki | = | 10.2 | nM | ALA2320210 | 7.99 | nM | Sus scrofa | ||
15. | ALA2315234 | 13.TFA , trans isomer | Ki | = | 18.1 | nM | ALA2320210 | 7.74 | nM | Sus scrofa | ||
16. | ALA2315235 | 14.TFA, cis isomer | Ki | = | 55 | nM | ALA2320210 | 7.26 | nM | Sus scrofa | ||
17. | ALA2315236 | 15.3TFA | Ki | = | 17.8 | nM | ALA2320210 | 7.75 | nM | Sus scrofa | ||
18. | ALA2315237 | 16.TFA | Ki | = | 41.7 | nM | ALA2320210 | 7.38 | nM | Sus scrofa | ||
19. | ALA2315238 | 17.TFA, cis isomer | Ki | = | 126 | nM | ALA2320210 | 6.90 | nM | Sus scrofa | ||
20. | ALA3325623 | 1 | INH | 0 | ALA3363614 | Active | % | Sus scrofa |