# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Carfilzomib | 2 | INH | 0 | ALA4003670 | Active | % | Mus musculus | ||||
2. | Carfilzomib | 2 | INH | 0 | ALA4003675 | Active | % | Mus musculus | ||||
3. | ALA4078056 | 43 | INH | 0 | ALA4003675 | Active | % | Mus musculus | ||||
4. | ALA4102324 | 42 | INH | 0 | ALA4003675 | Active | % | Mus musculus | ||||
5. | ALA4104744 | 39 | INH | > | 70 | % | ALA4003675 | % | Mus musculus | |||
6. | ALA4094582 | 36 | INH | 0 | ALA4003675 | Active | % | Mus musculus | ||||
7. | ALA4078693 | 35 | INH | > | 70 | % | ALA4003675 | % | Mus musculus | |||
8. | ALA4061262 | 30 | INH | > | 70 | % | ALA4003675 | % | Mus musculus | |||
9. | ALA4078056 | 43 | INH | 0 | ALA4003670 | Active | % | Mus musculus | ||||
10. | ALA4102324 | 42 | INH | 0 | ALA4003670 | Active | % | Mus musculus | ||||
11. | ALA4094582 | 36 | INH | 0 | ALA4003670 | Active | % | Mus musculus | ||||
12. | KZR-616 | ZETOMIPZOMIB | IC50 | = | 0.483 | uM | ALA4411754 | 6.32 | nM | Mus musculus | ||
13. | ALA4443505 | 3 | IC50 | = | 0.694 | uM | ALA4411754 | 6.16 | nM | Mus musculus | ||
14. | ALA4452892 | 10 | IC50 | = | 0.378 | uM | ALA4411754 | 6.42 | nM | Mus musculus | ||
15. | ALA4465456 | 2 | IC50 | = | 0.038 | uM | ALA4411754 | 7.42 | nM | Mus musculus | ||
16. | ALA4441524 | 1 | IC50 | = | 2.65 | uM | ALA4411754 | 5.58 | nM | Mus musculus | ||
17. | ALA4550864 | 7 | IC50 | = | 6.81 | uM | ALA4411754 | 5.17 | nM | Mus musculus | ||
18. | ALA4454809 | 6 | IC50 | = | 0.507 | uM | ALA4411754 | 6.29 | nM | Mus musculus | ||
19. | ALA4464640 | 5 | IC50 | = | 0.118 | uM | ALA4411754 | 6.93 | nM | Mus musculus | ||
20. | ALA3319584 | 18 | IC50 | = | 2.34 | uM | ALA4411754 | 5.63 | nM | Mus musculus |