# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5180795 | 54 | IC50 | > | 40 | uM | ALA5161725 | nM | Homo sapiens | |||
2. | ALA5183361 | 50 | IC50 | > | 40 | uM | ALA5161725 | nM | Homo sapiens | |||
3. | ALA5209480 | 31 | IC50 | > | 40 | uM | ALA5161725 | nM | Homo sapiens | |||
4. | M3258 | 50 | IC50 | > | 30000 | nM | ALA5151697 | nM | Homo sapiens | |||
5. | ALA5188533 | 4 | IC50 | = | 11 | nM | ALA5151697 | 7.96 | nM | Homo sapiens | ||
6. | Carfilzomib | 2 | IC50 | = | 69 | nM | ALA5151697 | 7.16 | nM | Homo sapiens | ||
7. | ALA5171825 | 2 | IC50 | = | 2.7 | nM | ALA5151697 | 8.57 | nM | Homo sapiens | ||
8. | Bortezomib (PS-341) | 15 | IC50 | = | 2.9 | nM | ALA5151697 | 8.54 | nM | Homo sapiens | ||
9. | ALA5177192 | 4 | IC50 | > | 50 | uM | ALA5133898 | nM | Homo sapiens | |||
10. | ALA5205926 | 2 | IC50 | > | 50 | uM | ALA5133898 | nM | Homo sapiens | |||
11. | ALA5180193 | 1 | IC50 | > | 50 | uM | ALA5133898 | nM | Homo sapiens | |||
12. | ALA4542139 | 23h | IC50 | > | 10000 | nM | ALA4413414 | nM | Homo sapiens | |||
13. | ALA4442152 | 23i | IC50 | > | 10000 | nM | ALA4413414 | nM | Homo sapiens | |||
14. | Bortezomib (PS-341) | 15 | IC50 | = | 3 | nM | ALA4413414 | 8.52 | nM | Homo sapiens | ||
15. | ALA4441524 | 1 | INH | 0 | ALA4411813 | Active | % | Homo sapiens | ||||
16. | ALA4100295 | 12; KZR-504 | INH | 0 | ALA4411810 | Active | % | Homo sapiens | ||||
17. | ALA4441524 | 1 | INH | 0 | ALA4411807 | Active | % | Homo sapiens | ||||
18. | ALA4452892 | 10 | INH | 0 | ALA4411804 | Active | % | Homo sapiens | ||||
19. | ONX-0914 | PR-957 | INH | 0 | ALA4411804 | Active | % | Homo sapiens | ||||
20. | KZR-616 | ZETOMIPZOMIB | IC50 | = | 0.131 | uM | ALA4411749 | 6.88 | nM | Homo sapiens |