| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4070633 | 1; CCT245232 | pIC50 | = | 7.36 | ALA4329880 | 7.36 | nM | Homo sapiens | |||
| 2. |  CCT251236 | 26 | pIC50 | = | 7.48 | ALA4329880 | 7.48 | nM | Homo sapiens | |||
| 3. |  ALA4091953 | 28 | INH | 0 | ALA4329881 | Not Active | % | Homo sapiens | ||||
| 4. |  GDC-0879 | 10, GDC-0879, AR00341677 | IC50 | > | 10 | uM | ALA4329880 | nM | Homo sapiens | |||
| 5. |  Dabrafenib | 7, GSK2118436 | IC50 | > | 10 | uM | ALA4329880 | nM | Homo sapiens | |||
| 6. |  RAF265 (CHIR-265) | CHIR-265/RAF-265 | IC50 | > | 10 | uM | ALA4329880 | nM | Homo sapiens | |||
| 7. |  TAK-632 | 8B, TAK-632 | IC50 | > | 10 | uM | ALA4329880 | nM | Homo sapiens | |||
| 8. |  AZ 628 | SID137275881 | IC50 | > | 10 | uM | ALA4329880 | nM | Homo sapiens | |||
| 9. |  Vemurafenib (PLX4032, RG7204) | VEMURAFENIB | IC50 | > | 10 | uM | ALA4329880 | nM | Homo sapiens | |||
| 10. |  ALA4473676 | 8; CCT363294 | IC50 | = | 0.033 | uM | ALA4329880 | 7.48 | nM | Homo sapiens | ||
| 11. |  PLX-4720 | PLX-4720 | IC50 | = | 0.67 | uM | ALA4329880 | 6.17 | nM | Homo sapiens | ||
| 12. | ALA4091953 | 28 | IC50 | > | 10 | uM | ALA4329880 | nM | Homo sapiens | |||
| 13. | CCT251236 | 26 | IC50 | = | 0.033 | uM | ALA4329880 | 7.48 | nM | Homo sapiens | ||
| 14. | ALA4070633 | 1; CCT245232 | IC50 | = | 0.044 | uM | ALA4329880 | 7.36 | nM | Homo sapiens | ||
| 15. | CCT251236 | 26 | Ki(app) | = | 0.028 | uM | ALA4001302 | 7.55 | nM | Homo sapiens | ||
| 16. | CCT251236 | 26 | AC50 | = | 1.5 | uM | ALA4001302 | 5.82 | nM | Homo sapiens | ||
| 17. |  ALA4096048 | 17 | Ki(app) | = | 0.19 | uM | ALA4001302 | 6.72 | nM | Homo sapiens | ||
| 18. | ALA4096048 | 17 | AC50 | = | 10 | uM | ALA4001302 | 5.00 | nM | Homo sapiens | ||
| 19. |  TPh A | TPh A, TriphenylA | Kd | = | 1700 | nM | ALA4001279 | 5.77 | nM | Homo sapiens | ||
| 20. | TPh A | TPh A, TriphenylA | pKd | = | 5.77 | ALA4001279 | 5.77 | nM | Homo sapiens |
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